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2-{2-[3-(morpholin-4-yl)azetidin-1-yl]-2-oxoethyl}-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
9-(2,6-dimethylpyridin-4-yl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
4-[(dimethylamino)methyl]-1-[3-(piperidin-4-ylmethyl)benzoyl]azepan-4-ol
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
1-[4-({4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
2-(dimethylamino)-2-(4-methylphenyl)-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]acetamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl (1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
4-{5-[(4-methoxyphenyl)methyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperazin-2-one
2-{[2-(1H-imidazol-1-yl)propanamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-({[(5-methyl-1,2-oxazol-3-yl)methyl]amino}methyl)piperidin-2-one
3-(2-{4-[4-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]piperidin-1-yl}-2-oxoethyl)-2,3-dihydro-1H-isoindol-1-one
propan-2-yl 2-chloro-5-(1-ethyl-3-methyl-1H-pyrazole-5-amido)benzoate
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[3-(methylsulfanyl)propyl]acetamide
4-hydroxy-N-methyl-2-(4-methylphenyl)-N-[1-(4-methylpyridin-2-yl)propan-2-yl]pyrimidine-5-carboxamide
1,1,1-trifluoro-3-({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)propan-2-ol
{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-3-(1H-pyrrol-1-yl)propan-1-one
(1R,3S)-3-(2-aminoethoxy)-7-(8-fluoroquinoline-2-carbonyl)-7-azaspiro[3.5]nonan-1-ol
4-{[4-(5-methylfuran-2-yl)phenyl]methyl}morpholine
3-[1-(5-chlorothiophene-2-carbonyl)piperidin-3-yl]-N-cyclopropylpropanamide
3-(2H-1,3-benzodioxol-5-yl)-5-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(4-methylpyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[3-(2-methoxyphenyl)-3-methylpentyl]pyrimidin-2-amine
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}ethan-1-one
3-chloro-5-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-(cyclopropylmethyl)-5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-[2-(4-ethylpiperazin-1-yl)-2,3-dihydro-1H-indene-2-carbonyl]-1,2-oxazinane
6-fluoro-2-(6-methoxy-2,6-dimethylheptyl)-1H-1,3-benzodiazole
(3R,4R)-1-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
[(4-fluoro-3-methoxyphenyl)methyl](methyl)[1-(pyridin-3-yl)ethyl]amine
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-(pyrimidin-4-ylmethyl)benzamide
4-(piperidin-1-yl)-1-[4-(pyridin-4-yl)pyrimidin-2-yl]piperidine-4-carboxamide
methyl 5-{2-[(4-methylphenyl)carbamoyl]acetyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-chloro-5-{1-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1H-1,2,3-triazol-4-yl}pyridine
1-{2-[2-(3,5-dimethyl-1-benzofuran-2-yl)-1H-imidazol-1-yl]ethyl}piperidin-4-ol
[(1-cyclopentylpiperidin-4-yl)methyl]({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})(pyridin-3-ylmethyl)amine
4-methyl-3-[3-(morpholin-4-ylmethyl)phenyl]-1,2-dihydroquinolin-2-one
1-(1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
N-(4-{[(2,3-dimethyl-1H-indol-5-yl)methyl]sulfamoyl}phenyl)acetamide
2-{1-[(5-methylpyrazin-2-yl)methyl]-1H-imidazol-2-yl}benzoic acid
5-methanesulfonyl-N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-methylpyrimidin-4-amine
4-[(6-ethylpyrimidin-4-yl)amino]-1-[2-(4-fluorophenyl)ethyl]pyrrolidin-2-one
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
N-[2-(pyrrolidin-1-yl)ethyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
4-{1-butyl-5-[1-(2-oxopyrrolidin-1-yl)ethyl]-1H-1,2,4-triazol-3-yl}benzamide
methyl 2-({1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)acetate
N-[2-(3-chlorophenyl)ethyl]-1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-(4-methoxyphenyl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)cyclopropane-1-carboxamide
4-{[2-(pyridin-3-yl)morpholin-4-yl]methyl}-1H-pyrazole-3-carboxylic acid