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3-[2-(piperidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1H-indazole
3-(2-methoxyphenyl)-1-{4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}propan-1-one
N-(pyridin-3-ylmethyl)-4-[5-(trifluoromethyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
3,3-diethyl-1-{[(2S,4S)-4-fluoro-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}pyrrolidin-2-yl]methyl}urea
(3S,4S)-4-[({[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]piperidin-3-ol
2-{[4-methyl-1-(thiophen-2-yl)-1H-1,3-benzodiazol-2-yl]methoxy}acetic acid
N-{1-oxaspiro[4.5]decan-3-yl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
2-(1-ethylpiperidin-4-yl)-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]acetamide
methyl 3-{[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}propanoate
[3-(hydroxymethyl)-1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl]methanol
4-(4-methyl-4H-1,2,4-triazol-3-yl)-1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine
methyl 3-[(3S,4R)-1-[(2-chloro-6-fluorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoate
2-(3-{[(1S,5R)-6-(cyclopropylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}phenoxy)acetamide
(3R,4S)-1-(oxan-4-yl)-4-(propan-2-yl)pyrrolidin-3-amine
(2E)-N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
2-methyl-1-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,3-benzodiazole
3,5,7-trimethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole-2-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-(3-methyl-1H-pyrazole-5-carbonyl)pyrrolidine-2-carboxamide
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}acetamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-(1-phenylcyclopropyl)-1H-pyrazole-3-carboxamide
methyl 5-[(1-methyl-1H-1,2,3-benzotriazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(1-ethyl-1H-pyrazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
8-methoxy-2-methyl-4-(2,3,6-trifluorobenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{2-[1-(morpholine-4-carbonyl)piperidin-2-yl]ethyl}phenol
(2S,4S)-4-amino-1-[(2-cyanophenyl)methyl]-N-ethylpyrrolidine-2-carboxamide
(4aS,8aR)-6-(1-methyl-1H-pyrazole-4-carbonyl)-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(ethyl)(2-methylprop-2-en-1-yl)amine
4-(2-methoxyphenoxy)-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
2-chloro-N-ethyl-4-({[(3S,4S)-4-hydroxy-1-(propan-2-yl)pyrrolidin-3-yl]carbamoyl}amino)benzamide
[3-(4-methyl-1,3-thiazol-5-yl)propyl](6-methylhept-5-en-2-yl)amine
9-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclobutanecarboxamide
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-(4-phenylbenzoyl)piperidine
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-4-(2-oxopyrrolidin-1-yl)benzamide
N-[3-(5-acetylpyridin-2-yl)phenyl]acetamide
4-{[2-(2-methylpropanamido)ethyl]sulfamoyl}-N-(propan-2-yl)benzamide
4-(1H-pyrazol-1-yl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-4-carboxylic acid
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2,6-dimethylquinoline-3-carboxamide
2-[9-(morpholine-2-carbonyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
2-[2-(1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperidin-2-yl)ethyl]pyridine
N-methyl-N-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2,3-dihydro-1H-inden-2-amine
N-[(1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}piperidin-3-yl)methyl]furan-2-carboxamide
1-[2-(piperazin-1-yl)ethyl]-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]-N-(2-methoxyethyl)-1-methyl-1H-1,3-benzodiazol-2-amine
3-methoxy-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)benzamide
3-(2H-1,3-benzodioxol-5-yl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}propan-1-one
1-{3-[(cyclopropylmethyl)amino]-5-(dimethylsulfamoyl)benzoyl}piperidine-3-carboxamide
N-benzyl-1-cyclopropyl-4-oxo-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,4-dihydropyridine-3-carboxamide
1-[5-(4-methoxyphenyl)-1H-1,3-benzodiazol-2-yl]ethan-1-ol
4-{[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]methyl}-N-methylbenzamide