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N5-cyclopentyl-N6-[2-(propan-2-yloxy)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
ethyl 3-{[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]amino}propanoate
N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)furan-2-carboxamide
2-{2-[4-(1-hydroxy-2-methylpropyl)piperidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
ethyl 1-[1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]piperidine-4-carboxylate
3-(3-fluorophenyl)-1-methyl-3-[2-oxo-2-(4-phenylazepan-1-yl)ethyl]pyrrolidine-2,5-dione
3-[(ethylcarbamoyl)methyl]-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
5-methanesulfonyl-1'-[(6-methylpyridin-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(4aR,7aS)-1-[2-(2,3-difluoro-4-methylphenoxy)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-(1-benzothiophen-2-ylmethyl)-3-[2-(dimethylamino)ethyl]-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]-3-propyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(4aS,7aR)-1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-amino-6-(2H-1,3-benzodioxol-5-yl)-4-[2-(propan-2-yl)pyrimidin-5-yl]pyridine-3-carbonitrile
1-(diethylamino)-3-[2-methoxy-5-({[(4-methoxyphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
1-(2-chloro-6-fluoro-3-methylbenzoyl)-3-(1-methyl-1H-imidazol-2-yl)piperidine
[(3R,4R)-1-[(6-fluoroquinolin-2-yl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-ethyl-5-[1-(3-methylpyridin-2-yl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]pyrimidine
4-(2-methylphenoxy)-1-(pyridine-4-carbonyl)piperidine-4-carboxylic acid
4-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-3-amine
2-(3-phenyl-1,2,4-oxadiazol-5-yl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-amino-1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
4-(5-{[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
2-(1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-4-yl)ethan-1-ol
N-(4-methoxy-2-methylphenyl)-3-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]propanamide
2-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}benzonitrile
1-[(2-fluorophenyl)methyl]-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-1H-1,2,3-triazole-4-carboxamide
4-[(4-fluorophenyl)methyl]-1-(4-methyl-1,3-thiazol-2-yl)piperidine
3-[(ethylamino)methyl]-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
1-[(1R,2R)-2-(benzyloxy)cyclopentyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
N-cyclopentyl-N'-[2-(2-ethoxyphenoxy)ethyl]-N'-methylethanediamide
3-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-methyl-1-(1,3,4-thiadiazol-2-yl)urea
5-{3-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-oxopropyl}-5-(thiophen-2-ylmethyl)pyrrolidin-2-one
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-methyl-N-(1,2-oxazol-5-ylmethyl)acetamide
2-({[(3R,4R)-1-[(2-chloro-4-fluorophenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-{[3-(4-methoxyphenyl)propanamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}acetamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}propanamide
1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-4-(pyrrolidine-1-carbonyl)piperidine
5-[4-(hydroxymethyl)piperidin-1-yl]-1-methyl-N-[(5-methylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(1H-1,2,4-triazol-3-ylsulfanyl)acetamide
1'-[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]spiro[indene-1,4'-piperidine]
1-{4-[({3-azaspiro[5.5]undecan-9-yl}amino)methyl]phenyl}pyrrolidin-2-one
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-1-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
ethyl 4-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-2-(methylsulfanyl)pyrimidine-5-carboxylate
(2S)-1-[4-(pyridin-4-yl)pyrimidin-2-yl]pyrrolidine-2-carboxylic acid
2-{4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-hydroxypyridine-3-carboxamide