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2-(methoxymethyl)-5-{[4-(3-methylphenoxy)piperidin-1-yl]methyl}pyrimidine
3,3-dimethyl-1-[(3S,4R)-1-[(3-methylthiophen-2-yl)sulfonyl]-4-(propan-2-yl)pyrrolidin-3-yl]urea
5-(2-fluorophenyl)-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1,2,4-triazin-3-amine
(2,1,3-benzoxadiazol-5-ylmethyl)({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
1-[3-(1H-imidazol-1-yl)propyl]-5-(3-methylphenyl)-4-phenyl-1H-imidazole
1-{1'-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
N-cyclopropyl-3,5-dimethoxy-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)benzamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
1-(1-methylpiperidin-4-yl)-N-(3-phenylpropyl)piperidine-3-carboxamide
(2S)-2-amino-2-(2-chlorophenyl)-N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
2-oxo-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-1,2-dihydroquinoline-4-carboxamide
4-[(diethylamino)methyl]-5-ethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]furan-2-carboxamide
1-(oxane-4-carbonyl)-4-(thiophene-2-carbonyl)piperazine
N-[(3R,5S)-5-(diethylcarbamoyl)-1-[3-(methylsulfanyl)propyl]pyrrolidin-3-yl]pyridine-3-carboxamide
5-tert-butyl-4-({3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)furan-2-carboxamide
2-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-2-oxo-N-phenylacetamide
2-{[(3-hydroxy-2-oxo-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]amino}-2-methylpropanamide
2-{[(cyclohex-3-en-1-ylmethyl)(methyl)amino]methyl}-3,4-dihydroquinazolin-4-one
1-(dimethyl-1,3-oxazole-4-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
(1S,6R)-9-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-3,9-diazabicyclo[4.2.1]nonan-4-one
1-({2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}sulfonyl)azepane
3-{[(2,2-dimethylpropyl)amino]methyl}-1-[(2-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
3-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]-1,2,3,4-tetrahydroisoquinolin-1-one
N-({7-[(4-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2,5-dimethylfuran-3-carboxamide
(1R,3S)-3-{[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]carbamoyl}cyclopentane-1-carboxylic acid
4-(azocane-1-carbonyl)-8-methyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
[(5-methoxy-1H-indol-2-yl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
3-[2-(4-fluorophenyl)ethyl]-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine
2-(4-ethoxyphenyl)-N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
2-(morpholin-2-yl)-N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)acetamide
5-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile
4-methoxy-2-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]phenol
3-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-(5-methyl-2,1,3-benzothiadiazol-4-yl)urea
4-[4-(pyrrolidine-1-carbonyl)phenoxy]-1-{[4-(trifluoromethyl)phenyl]methyl}piperidine
5-(morpholin-4-ylmethyl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]furan-3-carboxamide
4-{1-[4-(pyrimidin-2-yl)phenyl]ethyl}morpholine
4-[3-(cyclohexylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-(prop-2-en-1-yl)pyrrolidin-2-one
benzyl(methyl){[3-(4-propylpiperazine-1-carbonyl)-1,2-oxazol-5-yl]methyl}amine
3-{[(2H-1,3-benzodioxol-5-ylmethyl)(pyridin-3-ylmethyl)amino]methyl}pyrrolidin-3-ol
N-[(3R,4S)-1-(2-methylpyridin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-(2-oxopiperidin-1-yl)acetamide
1-(2,3-dihydro-1H-inden-2-yl)-4-(3-propyl-1H-pyrazole-4-carbonyl)-1,4-diazepane
2-({[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)amino)-1-phenylethan-1-ol
(3S,9aR)-8-[(3,4-dimethylphenyl)methyl]-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-methyl-4-{[4-(2-methylpropyl)-1,4-diazepan-1-yl]methyl}benzene-1-sulfonamide
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2,6-dimethylquinoline-4-carboxamide
(3aR,6aR)-2-(1-methyl-1H-pyrazole-3-carbonyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-[1-(4-chlorophenyl)cyclobutanecarbonyl]-N-(3-fluorophenyl)-6-azaspiro[2.5]octane-1-carboxamide
4-{2-[1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidin-2-yl]ethyl}phenol
(4aS,7aR)-1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-hydroxy-1-[(3-methylphenyl)methyl]-3-[(4-phenylpiperazin-1-yl)methyl]piperidin-2-one