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3-[(3R,4S)-4-(dimethylamino)-1-phenylmethanesulfonylpiperidin-3-yl]propanoic acid
3-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)-1-methyl-1,4-dihydroquinolin-4-one
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-1,2-oxazole-3-carboxamide
2-(2-hydroxyethyl)-8-[(2,3,6-trifluorophenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
[1-(2,1-benzoxazole-3-carbonyl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
(4aS,8aS)-2-[6-(dimethylamino)pyrazin-2-yl]-decahydro-2,7-naphthyridin-4a-ol
2-{[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazol-5-yl]formamido}acetic acid
2-(2-{[2-(methylsulfamoyl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-{2-methyl-1-[7-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]propyl}pyridine-2-carboxamide
1-{1-[3-(1-methylcyclopropyl)propanoyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
4-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)benzonitrile
2-amino-4-ethyl-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-1,3-thiazole-5-carboxamide
2-({1-[3-(methylcarbamoyl)phenyl]-1H-1,3-benzodiazol-2-yl}methoxy)acetic acid
3-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}piperazin-1-yl)-1,2-benzothiazole
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-2,1,3-benzoxadiazole-5-carboxamide
5-(dimethylamino)-2-[2-(6-methylpyridin-2-yl)ethyl]-2,3-dihydropyridazin-3-one
2-ethoxy-6-({[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amino}methyl)phenol
dimethyl({[1-(3-phenylprop-2-yn-1-yl)piperidin-3-yl]methyl}sulfamoyl)amine
7-cyclobutaneamido-1-methyl-2-(pyridin-4-yl)-N-[2-(thiophen-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
2-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
N-cyclohexyl-3-{[1-(propan-2-yl)-1H-pyrazol-4-yl]formamido}propanamide
2-[(3S,4R)-3-acetamido-4-(4-methylphenyl)pyrrolidin-1-yl]acetic acid
2,3,6-trimethyl-N-[2-(pyridin-3-yloxy)propyl]quinoline-4-carboxamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
7-cyclopentyl-2-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
[(2,6-difluoro-3-methoxyphenyl)methyl](2-methoxyethyl)(oxolan-2-ylmethyl)amine
4-{4-phenyl-1-[1-(pyridin-4-yl)propan-2-yl]-1H-imidazol-5-yl}-2-(propan-2-yl)pyrimidine
6-methyl-2-(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
N-(3-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}-2,5-dimethyl-1H-pyrrol-1-yl)acetamide
(2S,4S)-4-amino-N-ethyl-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]pyrrolidine-2-carboxamide
ethyl 4-[5-(3-fluoro-4-methoxyphenyl)-1,2,4-triazin-3-yl]piperazine-1-carboxylate
2-(3-methylbut-2-en-1-yl)-N-(2-methylphenyl)-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide
{2-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}urea
N-(1-{7-[(4-ethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
6-methyl-14-{2-[(propan-2-yl)amino]pyrimidin-5-yl}-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
(1S,5R)-6-propyl-3-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-methyl-N-(2-phenoxyethyl)acetamide
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
5-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid
N-(furan-2-ylmethyl)-1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-({[1-(5-methyl-1,3-benzoxazol-2-yl)piperidin-4-yl]amino}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-imidazol-4-ylmethyl)piperidine
N-{2-fluoro-5-[({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}carbamoyl)amino]phenyl}-2-methylpropanamide
3-(3-hydroxypropyl)-5-(3-phenylpropyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
(2R,6S)-2,6-dimethyl-4-(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)morpholine
1-[2-(3-fluorophenyl)ethyl]-4-(thiophen-2-ylmethyl)piperazine
5,6-dimethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-oxo-1,2-dihydropyridine-3-carboxamide