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2-methyl-4-(4-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}phenyl)butan-2-ol
N-{1-[1-(1-methoxypropan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
3-[methyl({3-[4-(4-methylphenyl)piperazin-1-yl]propyl})amino]-1λ6-thiolane-1,1-dione
2-[2-(1-cyclohexyl-2,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamido]-N-methylacetamide
N-{4-[1-(1-methoxybutan-2-yl)-4-phenyl-1H-imidazol-5-yl]phenyl}acetamide
methyl 2-(cyclopropylsulfamoyl)-6-[(4-methoxy-2,3-dimethylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-amine
N-[3-(1H-indazol-1-yl)propyl]-1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-[5-(7-hydroxy-6-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)furan-2-yl]benzonitrile
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(dimethyl-1,3-thiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-(2-methoxyphenyl)-N-[2-(1H-1,2,3-triazol-1-yl)ethyl]benzamide
3-{1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
2-(2-methoxyphenoxy)-N-{[1-(thian-4-yl)piperidin-3-yl]methyl}acetamide
N,5-dimethyl-N-(oxan-4-yl)-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
6-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(3,3-dimethylbutyl)-4-(2-hydroxyacetyl)-1,4-diazepane-6-carboxylic acid
2-methyl-1-{2-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-2-oxoethyl}-1,4-dihydroquinolin-4-one
(3R,4S)-4-cyclopropyl-1-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]pyrrolidin-3-amine
9-(3-phenylpropyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-({[(3R,4R)-1-[1-(4-fluorophenyl)cyclopropanecarbonyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-4-phenyl-5-(thiophen-2-yl)-1H-imidazole
2-amino-4-(3-methylthiophen-2-yl)-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(2-methyl-4-phenylpyrimidine-5-carbonyl)pyrrolidin-3-yl]methanol
2-[4-(2,5-dimethylfuran-3-carbonyl)morpholin-3-yl]-1-[4-(hydroxymethyl)piperidin-1-yl]ethan-1-one
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-[(2,4,5-trimethylphenyl)methyl]pyrrolidin-3-yl]methanol
N-[2-(cyclohexylsulfanyl)ethyl]-1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carboxamide
5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-N-(propan-2-yl)pyrimidin-2-amine
4-(1-{1-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperidin-4-yl}piperidine-4-carbonyl)morpholine
methyl (2S)-1-[2-(2-aminoethyl)quinazolin-4-yl]pyrrolidine-2-carboxylate
5-(2-benzyl-1,3-thiazole-4-carbonyl)-N-cyclopentyl-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[7-(hydroxymethyl)-9-(pyridin-4-yl)-3,9-diazaspiro[5.5]undecan-3-yl]acetic acid
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-3-ol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carboxamide
(2S,4S,5R)-4-[(1,3-dihydroxypropan-2-yl)carbamoyl]-2-ethyl-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
(3S,9aR)-8-(2,5-dimethylbenzenesulfonyl)-3-ethyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(3-ethoxypropyl)-2-[(3-fluorophenyl)methyl]-6-methyl-1-[3-(morpholin-4-yl)propyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(3-fluorophenyl)-4-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]-4-oxobutanamide
5-(2,5-dimethylfuran-3-yl)-N-[3-(pyridin-3-yl)propyl]-1,2,4-triazin-3-amine
5-methoxy-1-methyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1H-indole-2-carboxamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)pyrrolidine-3-carboxamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1-(3-hydroxyphenyl)-5-oxopyrrolidine-3-carboxamide
2-(2-{[benzyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxy)ethan-1-ol
8-fluoro-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}quinoline-2-carboxamide
5-{[5-(4-fluoro-2-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-1H-1,2,3,4-tetrazole
{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[2-(1H-imidazol-1-yl)ethyl]methylamine
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
N-({1-[(2-hydroxy-6-methoxyquinolin-3-yl)methyl]piperidin-3-yl}methyl)acetamide
(3S)-N,N-dimethyl-1-[(6-methylpyridin-2-yl)methyl]azepan-3-amine
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(5-methyl-1,3-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane