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3-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-6-methylpyridazine
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(3-phenylpropoxy)phenyl]acetamide
4,6-dimethyl-3-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1,2-dihydropyridin-2-one
4-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl](pyridin-3-yl)methyl}morpholine
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)propanamide
3-(azepane-1-sulfonyl)-N-(1,3-thiazol-2-ylmethyl)benzamide
N-[1-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-2-(2-fluorophenyl)ethyl]-N,2-dimethylfuran-3-carboxamide
(3S,7S,8aS)-7-{[(3,4-difluorophenyl)methyl]amino}-3-[(1R)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-3-cyclopropyl-1H-pyrazole-5-carboxamide
1-(3-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-oxopropyl)-6-methyl-1,2-dihydropyridin-2-one
2-({4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazin-1-yl}methyl)benzonitrile
2-[2-(4-benzylpiperidin-1-yl)-2-oxoethyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-5-methyl-N-[3-(methylsulfanyl)propyl]-1H-pyrazole-4-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidine-2-carboxamide
3-(azetidine-1-carbonyl)-N-ethyl-N-(oxan-2-ylmethyl)benzene-1-sulfonamide
5-(methoxymethyl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]furan-2-carboxamide
N-{[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-3-yl]methyl}-2-(4-methoxyphenyl)acetamide
N-[(3S,4R)-1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-{1-[3-(1H-1,2,4-triazol-1-yl)adamantane-1-carbonyl]azetidin-3-yl}pyridine
(2R,3R,6R)-3-(2,3-difluorophenyl)-N-ethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
5-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole
(4aS,7aR)-1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)-1-(pyridin-2-ylmethyl)piperidin-2-one
2-amino-6-(2H-1,3-benzodioxol-5-yl)-4-(furan-2-yl)pyridine-3-carbonitrile
N-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-N-methyloxan-4-amine
(4aS,8aR)-6-[1-(1H-imidazol-1-ylmethyl)cyclopropanecarbonyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2,2-dimethylpropyl 4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
3-cyano-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzamide
1-[1'-(4-ethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl)(oxolan-3-ylmethyl)amine
3-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
4-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]carbamoyl}amino)-N,3-dimethylbenzamide
4-(pyridin-2-yl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]pyrimidin-2-amine
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-(pyridine-3-carbonyl)piperidin-4-amine
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-3-amine
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[2-(1,3-thiazol-4-yl)ethyl]pyrimidine-5-carboxamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-(2-hydroxyphenyl)-N-methyl-N-[1-(pyridin-3-yl)pentyl]-1H-pyrazole-5-carboxamide
N-[(3-chlorophenyl)methyl]-2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
dimethyl(2-{[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amino}ethyl)amine
ethyl 1-ethyl-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
5-{[2-(2-acetamidoethyl)piperidin-1-yl]methyl}-2-hydroxybenzoic acid
4-[1-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)ethyl]-1,2-dihydrophthalazin-1-one
N-cyclopropyl-3-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}propanamide
1-[3-(2-methylphenyl)piperidin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
1-(3-carbamoylpyridin-2-yl)-4-(2-fluoro-5-methylphenoxy)piperidine-4-carboxylic acid
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)[(6-methylpyridin-2-yl)methyl]amine
(1-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)(phenyl)methanol
N-[(1R)-1-cyclohexylethyl]-5-oxo-1,4,9-triazaspiro[5.5]undecane-9-carboxamide