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(1S,5R)-6-(2-methoxyethyl)-3-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
N-ethyl-N-methyl-2-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-amine
N-(furan-3-ylmethyl)-N-methyl-3-{[(2S)-pyrrolidin-2-ylmethyl]sulfamoyl}benzamide
2-{3-[2-amino-3-cyano-6-(propan-2-yl)pyridin-4-yl]phenoxy}acetamide
5,6-dimethyl-2-[3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carbonitrile
N-[(3S,4R)-1-{2-methylimidazo[1,2-a]pyridine-3-carbonyl}-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
5-(oxolane-2-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-cyclohexyl-3-methyl-5-(2H-1,2,3-triazol-2-ylmethyl)-1H-1,2,4-triazole
N-[(3S,4R)-1-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-4-propylpyrrolidin-3-yl]acetamide
2-amino-3-ethyl-N-[2-(quinolin-8-yloxy)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
6-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-{1-methyl-4-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]piperazin-2-yl}ethan-1-ol
2-methyl-5-(3-methyl-1H-1,2,4-triazol-5-yl)pyrazine
6-ethyl-1-methyl-N-[1-(thiophen-2-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-{methyl[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}propane-1,2-diol
{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
1-cyclopentyl-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxamide
4-{[1-(2-methoxyphenyl)-5-(2-methyloxolan-2-yl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
2-[2-(propan-2-yloxy)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-{1-[2-(3-chloro-4-fluorophenyl)-1H-imidazol-1-yl]ethyl}-5-methylpyridine
(4aS,7aS)-6-(5-methyl-2-phenylfuran-3-carbonyl)-octahydro-1H-pyrrolo[3,4-b]pyridine
2-({[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
N-ethyl-1-methyl-N-(2-methylprop-2-en-1-yl)-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-(1H-imidazol-1-ylmethyl)piperidine
3-{2-[4-(2,3-dimethylphenyl)piperazin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
5-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
ethyl 1-[2-(dimethylamino)ethyl]-5-[(3-hydroxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
5-methyl-2-(2-methylpropanamido)-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]benzamide
2-ethoxy-N-[(4-methoxyphenyl)methyl]-N-[(3-methylphenyl)methyl]acetamide
(3R,7S,8aS)-7-[({3-[(diethylamino)methyl]-4-methoxyphenyl}methyl)amino]-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(3S,4R)-4-(3-fluorophenyl)-1-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]pyrrolidine-3-carboxylic acid
N-[(4,6-dimethylpyridin-3-yl)methyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
3-chloro-4-fluoro-N-[(3S)-2-oxoazepan-3-yl]-1-benzothiophene-2-carboxamide
1-(3-chlorophenyl)-4-[1-(3-ethynylbenzoyl)piperidin-3-yl]piperazine
3-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}benzoic acid
N-({6-methyl-2-[methyl(1H-pyrazol-5-ylmethyl)amino]quinolin-3-yl}methyl)-N-(oxolan-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(quinoxalin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3R,4R)-4-(azepan-1-yl)-1-[1-(2,3-dimethylphenyl)piperidin-4-yl]piperidin-3-ol
N-[2-(3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)propyl]pyridine-2-carboxamide
N-{5-[2-(2-hydroxyphenoxy)acetamido]-2-methoxyphenyl}pentanamide
1-[6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carbonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
(1R,5S,6R)-3-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-[2-(1H-pyrazol-1-yl)ethyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
4-chloro-N-{5H,6H,7H,8H,9H,10H-cyclohepta[b]indol-2-ylmethyl}-1-methyl-1H-pyrazole-5-carboxamide
(3S,4S)-1-(2-aminopyridine-4-carbonyl)-4-(2H-1,3-benzodioxol-5-yl)piperidin-3-ol
3-{4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl}azepan-2-one
5-(2-chloro-4-methoxyphenoxymethyl)-N-(1H-imidazol-2-ylmethyl)-N-methyl-1H-pyrazole-3-carboxamide
[(3aS,6aS)-2-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
ethyl (4aS,8aR)-6-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-decahydro-1,6-naphthyridine-4a-carboxylate