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8-fluoro-2-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]quinoline
N,2-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4-phenyl-1,3-thiazole-5-carboxamide
2-[3-oxo-9-(4-phenylbutanoyl)-2,9-diazaspiro[5.5]undecan-2-yl]acetic acid
4-(3-methyl-1,2,4-oxadiazol-5-yl)-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-(1-methyl-1H-pyrazol-5-yl)-N-(propan-2-yl)propanamide
N-methyl-4-(1-methyl-1H-pyrazol-4-yl)-N-[2-(morpholin-4-yl)ethyl]pyrimidin-2-amine
3-({[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
2-[4-(furan-3-ylmethyl)morpholin-3-yl]-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]acetamide
4-chloro-2-({4-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)phenol
1-[2-methyl-3-(1H-pyrazol-1-yl)propanoyl]-4-phenoxypiperidine-4-carboxylic acid
2-hydroxy-N-[(3R,5S)-1-(1H-imidazol-2-ylmethyl)-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]pyridine-3-carboxamide
5,6-dimethyl-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-{1-[2-(methylsulfanyl)acetyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
5-acetyl-6-methyl-3-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
1-(2-{[3-(1H-imidazol-1-yl)propyl]amino}-4-methylpyrimidin-5-yl)ethan-1-one
1,9-dimethyl-4-[(3-methylquinoxalin-2-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(2-aminoethyl)-N-cyclopropyl-N-[(3-methylthiophen-2-yl)methyl]quinazolin-4-amine
N,2,6-trimethyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)quinoline-4-carboxamide
1-(3-chlorophenyl)-4-[1-(2-methoxypyridine-3-carbonyl)piperidin-3-yl]piperazine
1-[3-(3-methylphenoxy)azetidin-1-yl]-3-(1-methylpiperidin-2-yl)propan-1-one
{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(trifluoromethyl)phenyl]methyl}amine
N-methyl-3-(morpholine-4-carbonyl)-N-(oxolan-3-ylmethyl)benzene-1-sulfonamide
1-[(4-ethyl-1,3-thiazol-2-yl)methyl]-4-[2-(methylsulfanyl)propyl]-1H-1,2,3-triazole
{[2-(furan-2-yl)pyrimidin-5-yl]methyl}(methyl)[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]amine
5-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1H-pyrazol-3-yl]-1-(2-fluorophenyl)-3-methyl-1H-1,2,4-triazole
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl](methyl){[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
3-[(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)methyl]-2,3-dihydro-1H-isoindol-1-one
N-(2-ethoxyethyl)-3-{[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]sulfamoyl}benzamide
N-(1-{1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
2-fluoro-N-{3-[3-(2-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl}benzamide
3-{[9-(furan-3-ylmethyl)-7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]methyl}phenol
1-(cyclohex-3-en-1-ylmethyl)-3-[4-(3,4-difluorophenyl)-1H-pyrazol-5-yl]piperidine
N-[1-({4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}methyl)piperidin-4-yl]acetamide
4-[5-(1,4-dioxan-2-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]-2-methylpyridine
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
2-butyl-8-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(4-benzyl-1H-pyrazol-5-yl)-1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]piperidine
2-methyl-8-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
4-[(3-fluorophenyl)methyl]-1-(4-phenylbutan-2-yl)-1,4-diazepan-5-one
1-[(2,3-dichlorophenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-[4-(5-phenylthiophen-2-yl)-1H-pyrazol-1-yl]acetamide
1-(1H-imidazol-2-ylmethyl)-4-(piperidin-1-ylmethyl)piperidine
8-(2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
2-({[2-(2-ethyl-1H-imidazol-1-yl)ethyl]amino}methyl)-6-methylquinolin-4-ol
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-amino-4-(3,4-dihydroxyphenyl)-6-(2,5-dimethoxyphenyl)pyridine-3-carbonitrile
N-cyclopropyl-5-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-(2-methylphenyl)-N-[2-(morpholin-4-yl)ethyl]-3-phenylpropanamide
6-{[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one