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N-(propan-2-yl)-1-[(1s,4s)-4-[(2E)-3-(4-methoxyphenyl)prop-2-enamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
7-(5-chloropyridin-2-yl)-4-[(1-ethyl-1H-imidazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 1-(3-{4-[(benzylamino)methyl]phenoxy}-2-hydroxypropyl)piperidine-4-carboxylate
[(1-cyclopentylpiperidin-4-yl)methyl][(2,4-dimethoxyphenyl)methyl](oxolan-2-ylmethyl)amine
N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-[4-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
1-(furan-3-carbonyl)-4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-1,4-diazepane
2-[1-(3-methylbut-2-en-1-yl)piperazin-2-yl]ethan-1-ol
(3S,4R)-1-(1,4-dithiepan-6-yl)-4-phenylpyrrolidine-3-carboxylic acid
N-phenyl-5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)pyrimidin-2-amine
1-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
11-(6-chloro-2-fluoro-3-methoxyphenyl)-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
[2-(isoquinolin-5-yl)-1,3-thiazol-4-yl]methanol
4-(1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)morpholine
2-methyl-5-(4-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}phenyl)-1,3,4-oxadiazole
(1S,5R)-3-[2-(2,3-dimethoxyphenyl)acetyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl (2S,4S,5R)-4-[(dicyclopropylmethyl)carbamoyl]-5-(2-fluorophenyl)-1-methylpyrrolidine-2-carboxylate
[(3R,4R)-1-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
2-[(4-chlorophenyl)methyl]-8-(1H-imidazol-4-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
6-methyl-2-oxo-N-[2-(pyridin-3-yloxy)propyl]-1,2-dihydropyridine-4-carboxamide
4-hydroxy-2-{[2-(2-methylphenyl)pyrrolidin-1-yl]methyl}quinoline-6-carboxamide
3-chloro-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,6-dimethylpyrazolo[1,5-a]pyrimidine-2-carboxamide
2-hydroxy-N-{2-[1-(pyridin-3-ylmethyl)piperidin-3-yl]ethyl}benzamide
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]acetamide
N-{[4-(but-2-yn-1-yloxy)-3-methoxyphenyl]methyl}-5-chloro-2-methoxy-N-(oxolan-2-ylmethyl)benzene-1-sulfonamide
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-3-phenyl-1,2-oxazole-4-carboxamide
3-{[4-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)piperidin-1-yl]methyl}phenol
1-methanesulfonyl-3-[2-(3-methoxyphenyl)ethyl]piperidine
1-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidine-3-carboxamide
N-(1-{1-[(2E)-3-(3,4-difluorophenyl)prop-2-enoyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylcyclopropanecarboxamide
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-4-(1H-1,2,4-triazol-5-yl)benzamide
5-(3-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-3-oxopropyl)-5-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-2-one
(2R,6R)-10-methoxy-4-[2-(thiophen-3-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-(4-methoxyphenoxymethyl)-4-(1,2-oxazolidine-2-carbonyl)-1,3-oxazole
3-{[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]methyl}benzonitrile
N-methyl-5-[(methylsulfanyl)methyl]-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}pyridin-2-amine
N,N-dimethyl-6-(3-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridazin-3-amine
N-[(1R,3S)-3-{[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)carbamoyl}cyclopentyl]-1-methyl-1H-pyrrole-2-carboxamide
(4-methyl-5-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methanol
2-[4-({methyl[(6-methylpyridin-2-yl)methyl]amino}methyl)phenyl]-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-4-one
2-(4-ethylpiperazin-1-yl)-N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]acetamide
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
2-{4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
1-(butan-2-yl)-N-ethyl-4-oxo-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,4-dihydropyridine-3-carboxamide
1-(2-methylpropyl)-5-[(pyridin-2-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}azepan-4-amine
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-2-(3-hydroxyadamantan-1-yl)acetamide
N-[(1-benzylpyrrolidin-3-yl)methyl]-5-(4-fluorophenyl)-1,2,4-triazin-3-amine
7-(2-methoxyphenyl)-2-(pyridin-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-{3-[3-(4H-1,2,4-triazol-4-yl)phenyl]phenyl}acetamide