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7-[(2S)-4,4-difluoropyrrolidine-2-carbonyl]-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(1S,5R)-6-(2-methoxyethyl)-3-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[ethyl({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]-1λ6-thiolane-1,1-dione
ethyl 1-methanesulfonyl-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
5-(2-chlorophenyl)-N-(2-oxopyrrolidin-3-yl)furan-2-carboxamide
2-{9-[3-(dimethylamino)benzoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
4-(4-fluorophenyl)-1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-1,2,3,6-tetrahydropyridine
N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)-4-(1H-pyrrol-1-yl)benzamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)quinoxaline-5-carboxamide
3-(4-chloro-1H-pyrazol-1-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]propan-1-one
4-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}-1,4-diazepane-1-carbaldehyde
2-(2,4-dichlorophenoxy)-1-[3-(hydroxymethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N-(1,2,4-thiadiazol-5-yl)benzamide
4-(4-benzyl-1H-1,2,3-triazol-1-yl)-N-(4-fluorophenyl)piperidine-1-carboxamide
2-oxo-6-phenyl-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,2-dihydropyridine-3-carboxamide
(3S,4S)-4-(3-methoxyphenyl)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-ol
8-(prop-2-ene-1-sulfonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
7-(3-methoxyphenyl)-2-(1-propyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-chloro-3-{1-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-imidazol-2-yl}-1-methyl-1H-indazole
N-[(1R,3S)-3-[(4-chlorophenyl)carbamoyl]cyclopentyl]-4-methylpiperazine-1-carboxamide
ethyl 5-{[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]methyl}-1-(4-methoxyphenyl)-1H-pyrazole-4-carboxylate
2-(methoxymethyl)-5-[(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)methyl]pyrimidine
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)[(4-methyl-1H-imidazol-5-yl)methyl]amine
2-(3-methylbut-2-en-1-yl)-8-(oxan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
1-(4-chlorophenyl)-N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)cyclopropane-1-carboxamide
2-(dimethylamino)-N-[3-({[1-(1-methyl-1H-pyrazol-5-yl)propyl]carbamoyl}amino)phenyl]acetamide
1-{2-[(2-methoxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1,4-diazepan-5-one
{8-methyl-2-[3-(piperidin-1-ylmethyl)piperidin-1-yl]quinolin-3-yl}methanol
(2S,4R)-4-amino-N-methyl-1-[2-(morpholin-4-yl)pyridine-3-carbonyl]pyrrolidine-2-carboxamide
1-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}urea
4-({2-[1-(5-methoxyfuran-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
1-ethyl-4-{[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
1-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]azepane
N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]pyrazolo[1,5-a]pyridine-7-carboxamide
N-[(5-chlorothiophen-2-yl)methyl]-2-(4-ethoxyphenyl)acetamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzamide
1-[2-(3,3-diphenylpiperidin-1-yl)-2-oxoethyl]-1,2-dihydropyridin-2-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)cyclohexanecarboxamide
N,5,7-trimethyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}pyrido[2,3-d]pyrimidin-4-amine
4-ethyl-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-5-methylthiophene-3-carboxamide
N-[(2,5-difluorophenyl)methyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
[3-benzyl-1-(1H-indol-2-ylmethyl)piperidin-3-yl]methanol
4-(3-hydroxy-3-methylbutyl)-N-{[(1r,4r)-4-carbamoylcyclohexyl]methyl}benzamide
1-[7-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3-phenylpiperidin-1-yl)ethan-1-one
N-cyclopropyl-N-({4-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-3-methylthiophene-2-carboxamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-decahydro-1,6-naphthyridin-2-one
[(4-methanesulfonylphenyl)methyl](methyl)[1-(pyridin-2-yl)ethyl]amine
4,6,7-trimethyl-2-{4-[1-(2-phenylethyl)piperidin-4-yl]-1,4-diazepan-1-yl}quinazoline
(1S,5R)-6-methyl-3-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclooctyl-2-[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]acetamide