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6-(3-chlorophenyl)-N-(2-hydroxypropyl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N2-(2-methoxyethyl)-N4-methyl-N4-[(1-methyl-1H-imidazol-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-[(3R,4S)-1-(cyclobutylmethyl)-4-phenylpyrrolidin-3-yl]-3-hydroxypropanamide
(3S,4S)-1-({3-methoxy-4-[(3-methylphenyl)methoxy]phenyl}methyl)piperidine-3,4-diol
1-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(pyridin-2-yl)ethan-1-one
(3S)-3-ethyl-4-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]morpholine
4-(3-hydroxy-3-methylbutyl)-N-[1-(thian-4-yl)piperidin-4-yl]benzamide
N,1-dimethyl-N-{[3-(methylsulfanyl)phenyl]methyl}azepane-2-carboxamide
1,4,6-trimethyl-3-[3-(2-phenylethyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-[4-(2H-1,3-benzodioxol-5-yl)-3,5-dimethyl-1H-pyrazol-1-yl]-N-[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]acetamide
4-(2-{1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]piperidin-2-yl}ethyl)morpholine
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-(4-chlorophenyl)-N-methyl-3-phenyl-N-(pyrazin-2-ylmethyl)propanamide
4-[5-(2-chlorophenyl)furan-2-amido]oxane-4-carboxylic acid
5-(4-cyclohexylphenyl)-N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1,2,4-triazin-3-amine
4-(morpholin-4-yl)-6-[(1E)-pent-1-en-1-yl]pyrimidin-2-amine
1-cyclopentyl-4-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
8-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(1R,5R)-6-(1H-indole-6-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
3-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-4-yl}-1,3-oxazolidin-2-one
N-(1-{7-[(3-ethoxy-2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
1-[2-(4-fluorophenoxy)ethyl]-4-phenyl-5-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazole
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-{1-[(dimethylcarbamoyl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[2-(pyridin-3-yl)ethyl]benzamide
1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propan-1-one
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
1-(5-methyl-1,2-oxazole-4-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
5-{2-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-1-(3-methoxypiperidin-1-yl)propan-1-one
(1R,2S,9R)-11-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
5-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-methyl-2-[(5-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carbonyl}pyridin-2-yl)amino]acetamide
N-methyl-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
N-ethyl-6-oxo-1-[2-(pyridin-2-yl)ethyl]-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-[(2-ethylpyrimidin-5-yl)methyl]-8-(quinolin-6-yl)-1,8-diazaspiro[4.5]decane
4-({[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)-6,8-dimethyl-2H-chromen-2-one
1-[(4-methoxyphenyl)methyl]-N-[2-(4-phenylpiperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-2-(phenylamino)pyrimidine-5-carboxamide
1-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(1,3-thiazol-4-yl)ethan-1-one
3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}propan-1-one
(1R,9S)-5-amino-3-(2,5-dimethoxyphenyl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
(2S,4S)-1-[2-(adamantan-1-ylsulfanyl)acetyl]-4-amino-N-methylpyrrolidine-2-carboxamide
6-ethyl-4-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)-1,2-dihydropyridin-2-one
1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-(oxolane-2-carbonyl)piperazine
N5-cyclopentyl-N6-[1-(pyridin-4-yl)propyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4-[5-(1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
3-methoxy-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)propanamide