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N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-4-yl)propanamide
3-{[1-(2-oxo-2-phenylacetyl)piperidin-4-yl]methyl}benzoic acid
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-(2-phenylethyl)piperidine-3-carboxamide
N-methyl-5-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
N-butyl-3,5-difluoro-N-(furan-2-ylmethyl)pyridine-2-carboxamide
N-butyl-N-[(2-fluorophenyl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-[(1-cyclopentanecarbonylpiperidin-3-yl)methyl]-3,5-dimethoxybenzamide
N-[2-(7-{[3-(furan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-methylpropanamide
5-phenyl-N-[4-(4-{[2-(1H-pyrazol-1-yl)ethyl]amino}piperidin-1-yl)phenyl]pentanamide
(3R,4R)-4-(hydroxymethyl)-1-[2-(4-methylphenoxymethyl)furan-3-carbonyl]piperidin-3-ol
N-(1-phenylbutyl)thiophene-3-carboxamide
3-{[1-(2-methoxyethyl)-3-(4-methyl-1,4-diazepane-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2-methyl-1H-indole
2-amino-6-(furan-2-ylmethyl)-4-(1H-indol-5-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]-4-[1-(5-phenoxyfuran-2-carbonyl)piperidin-3-yl]pyrimidine
3-[1-(1-benzofuran-2-carbonyl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
1-(5-methyl-1,2,4-oxadiazol-3-yl)-4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine
4-ethyl-N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-2-methyl-1,3-thiazole-5-carboxamide
N-cyclopropyl-3-({1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
5-[1-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)ethoxy]-3,4,7-trimethyl-2H-chromen-2-one
(2,1,3-benzoxadiazol-4-ylmethyl)[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-4-oxo-4H-chromene-3-carboxamide
1-[(3-methylpyridin-2-yl)methyl]-4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperazine
4,4,4-trifluoro-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
2-oxo-4-(piperidin-4-yl)-7-(pyrrolidin-1-yl)-1,2,3,4-tetrahydroquinoline-6-carboxamide
1-(4-{[1-(3-methylpyridin-2-yl)ethyl]amino}piperidin-1-yl)butan-1-one
2-{4-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]morpholin-3-yl}acetic acid
N-(oxolan-2-ylmethyl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-({1-[(3-ethenylphenyl)methyl]pyrrolidin-3-yl}methyl)-6-oxo-1,6-dihydropyridazine-3-carboxamide
2-{2-[(3,4-dihydro-2H-1-benzopyran-3-yl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
1-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}cyclopropane-1-carboxamide
(1R,9aR)-1-{[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-octahydro-1H-quinolizin-1-ol
4-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-6-(propan-2-yloxy)pyrimidin-2-amine
2-(ethanesulfonyl)-5-{[3-(2-fluorophenyl)pyrrolidin-1-yl]methyl}-1-(2-phenylethyl)-1H-imidazole
6-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
(3S,4R)-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-phenylpyrrolidine-3-carboxylic acid
2-{[2-(1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-hydroxy-4-(methylsulfanyl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}butan-1-one
3-[1-(6-methoxy-3-methyl-1-benzofuran-2-yl)-N-methylformamido]-N-methylbutanamide
5-ethyl-2-methyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrimidin-4-amine
{1-[(2-ethylpyrimidin-4-yl)methyl]piperidin-4-yl}(pyridin-2-yl)methanol
5-ethyl-3-[(2-ethyl-1,3-thiazol-4-yl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
4-[(dimethylamino)methyl]-1-[4-(1H-pyrrol-1-yl)benzoyl]azepan-4-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-ol
1-{2-[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]-2-oxoethyl}-4,4-dimethylpyrrolidin-2-one
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-carboxamide
[(3R,4S)-1-(1-benzofuran-5-ylmethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
4-{[4-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazol-1-yl]methyl}-1H-indole
1-{2-[6-(4-methyl-1H-pyrazol-1-yl)pyrimidin-4-yl]phenyl}ethan-1-one