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2-butyl-8-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[1-(furan-3-ylmethyl)-4-[2-(methylamino)pyridine-3-carbonyl]piperazin-2-yl]ethan-1-ol
4-(6-methyl-2-phenylpyrimidin-4-yl)-2-(trifluoromethyl)morpholine
N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N,2,6-trimethylquinoline-3-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-N-methylpiperidin-3-amine
(3R,5S)-N-[3-(1H-imidazol-2-yl)propyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
1-[(2,3-dimethoxyphenyl)methyl]-4-[(dimethylamino)methyl]azepan-4-ol
6-methyl-2-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
5-(2-ethoxybenzoyl)-1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
3-{[1-(oxane-2-carbonyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-4-oxo-1,4-dihydroquinoline-2-carboxamide
2-(2-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-pyrrol-1-yl)pyridine
3-({[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]carbamoyl}amino)-N-cyclopropyl-4-methoxybenzamide
5-{[(2-chloro-6-fluorophenyl)methyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(3R,4S)-4-(4-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-1-yl)oxolan-3-ol
1-{3-[5-(oxan-4-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyrrolidin-2-one
(1R,5S,6R)-6-{[(2-methoxyethyl)(1,3-thiazol-2-ylmethyl)amino]methyl}-N,N-dimethyl-3-azabicyclo[3.1.0]hexane-3-carboxamide
4-(4-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
8-(2-methoxy-6-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N,N-dimethyl-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}aniline
1-[(2-ethylpyrimidin-5-yl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-3-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-yl}urea
3-[1-(6-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)piperidin-3-yl]benzoic acid
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1H-indole
4-methyl-2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]quinoline
2-[2-methoxy-4-(thiomorpholin-4-ylmethyl)phenoxy]-1-(morpholin-4-yl)ethan-1-one
2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}ethan-1-one
6-(methoxymethyl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]pyrimidin-4-amine
N-cyclopropyl-1-(2,8-dimethylquinoline-3-carbonyl)piperazine-2-carboxamide
(1R,5S,8S)-3-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-8-methoxy-3-azabicyclo[3.2.1]octane
(3S,4S)-3-hydroxy-N-[3-(piperidine-1-carbonyl)phenyl]-4-(pyrrolidin-1-yl)pyrrolidine-1-carboxamide
4-(1,3-dimethyl-1H-pyrazol-5-yl)-3-[1-(pyrrolidin-1-yl)ethyl]-4H-1,2,4-triazole
4-{[(2-amino-5-ethyl-6-methylpyrimidin-4-yl)amino]methyl}-1-methyl-1,2,3,4-tetrahydroquinolin-2-one
5-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-N,N-dimethylpyridin-2-amine
2-(adamantan-1-yl)-4-hydroxy-N-[2-(pyridin-4-yl)ethyl]pyrimidine-5-carboxamide
1-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
N-ethyl-2-(4-{[4-(pyridin-2-yl)phenyl]methyl}piperazin-1-yl)acetamide
4-[2-fluoro-6-(propan-2-yloxy)phenyl]thiophene-2-carboxamide
(2S,4S)-4-amino-N-ethyl-1-[2-(1H-pyrazol-1-yl)benzoyl]pyrrolidine-2-carboxamide
8-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{4-[3-(3-methylphenyl)piperidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
N-[3-(3-benzyl-1H-1,2,4-triazol-5-yl)adamantan-1-yl](methylsulfanyl)formamide
1-[1-(isoquinolin-1-yl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
4-[2-(ethylcarbamoyl)phenyl]benzoic acid
4-(3-cyclopropyl-5-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,4-triazol-1-yl)-1-methylpiperidine
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-2-(5-fluoro-2-methyl-1H-indol-3-yl)acetamide
1-(4-chloro-2-methoxybenzoyl)-4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine
N-(5-methyl-1,2-oxazol-3-yl)-2-(4-methylpyrimidine-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-{2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid