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5-{imidazo[1,2-a]pyridine-2-carbonyl}-2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)acetamide
2-{[2-amino-6-(5-fluoroquinolin-8-yl)pyrimidin-4-yl]amino}ethan-1-ol
{3-[(3-chlorophenyl)methyl]-1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidin-3-yl}methanol
5-methyl-N-[3-(morpholin-4-yl)propyl]-6-(piperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
1-[2-(4-chlorophenyl)ethyl]-N-methyl-6-oxo-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
1-benzyl-4-[(4-cyclopentylpyrimidin-2-yl)amino]pyrrolidin-2-one
{3-[(2,4-difluorophenyl)methyl]-1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-3-yl}methanol
2-[1-(2-phenylethyl)-4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperazin-2-yl]ethan-1-ol
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)acetamide
1-benzyl-4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1H-pyrazole
(1S,5R)-N-(2-methoxyphenyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
5-ethyl-2-methyl-4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
N-benzyl-N-methyl-3-({methyl[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
N-({7-[2-(2-chlorophenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
3-methyl-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-phenylpiperidine
(2S,4R)-4-amino-1-[2-(3,4-dimethoxyphenyl)acetyl]-N,N-diethylpyrrolidine-2-carboxamide
4-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-N-(prop-2-en-1-yl)aniline
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-4-methylpiperazine-2-carboxamide
1-(6-chloropyridin-3-yl)-3-cyclopropyl-3-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
4-(propan-2-yl)-6-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrimidin-2-amine
2-cyclopentanecarbonyl-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-2-[(prop-2-en-1-yl)amino]benzamide
4-amino-N-(butan-2-yl)-N-[(3-methylthiophen-2-yl)methyl]pyridine-2-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-methyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}acetamide
1-cyclohexyl-4-[4-(3-hydroxy-3-methylbutyl)benzoyl]piperazin-2-one
2-(2H-1,3-benzodioxol-5-yloxy)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
(3S,4S)-1-[(2-methyl-1-benzothiophen-3-yl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
2-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-6-methylpyridine-3-carboxylic acid
6-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]-1,3-benzothiazole
1-(1-methylpiperidin-4-yl)-3-(4-phenoxybenzoyl)piperidine
1-(1-benzofuran-2-ylmethyl)-2-(5-methyl-1,2-oxazol-3-yl)piperidine
1-(2-chlorophenyl)-3-{1-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
benzyl({1-[1-(pyrimidin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)amine
1-[2-(cyclohex-1-en-1-yl)ethyl]-1-(cyclopropylmethyl)-3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
2-(4-{4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}quinazolin-2-yl)ethan-1-amine
6-[3-(1H-indazol-1-yl)propyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-{4-[4-(3-hydroxyphenyl)piperidine-1-carbonyl]piperidin-1-yl}-2-methoxyethan-1-one
8-[(2R)-oxolane-2-carbonyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
2-(4-{[butyl(pyridin-4-ylmethyl)carbamoyl]amino}phenyl)-N-methylacetamide
methyl 6-(7-hydroxy-6-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)pyridine-2-carboxylate
[(5-fluoro-1H-indol-2-yl)methyl](methyl){[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
1-ethyl-3-({5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-6-methyl-1,2-dihydropyridin-2-one
1-(3,5-difluorophenyl)-N-[(8-methoxy-2H-chromen-3-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)-4-(2-methylphenoxy)piperidine
(1r,4r)-4-[({4-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)amino]cyclohexan-1-ol
(3S,4R)-4-(2-methylphenyl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]pyrrolidine-3-carboxylic acid
3-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-1-methyl-1-[1-(4-methylpyridin-2-yl)propan-2-yl]urea
4-(3-fluorophenoxy)-1-(thiophene-3-carbonyl)piperidine
4-(6-chloro-1,3-benzothiazol-2-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol