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4-{[4-(oxan-4-yl)piperazin-1-yl]methyl}quinoline
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(trifluoromethyl)benzamide
1-(2-chloro-4,6-dimethylphenyl)-3-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}urea
7-(3-chloro-5-fluorobenzoyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-methyl-2-(morpholin-4-yl)propan-1-one
(3S,4R)-1-{2-[methyl(1-methylpiperidin-4-yl)amino]acetyl}-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
methyl 4-({ethyl[2-(1H-pyrazol-1-yl)ethyl]carbamoyl}amino)-3-methylbenzoate
4-ethoxy-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-2-amine
N-[3-(5-chloro-1H-1,3-benzodiazol-2-yl)propyl]-1-(4-fluorophenyl)cyclopropane-1-carboxamide
5-fluoro-N,N-dimethyl-2-[2-(morpholin-4-ylmethyl)phenyl]pyrimidin-4-amine
5-[(4-benzylpiperidin-1-yl)methyl]-N-methyl-N-[1-(pyridin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
(3aR,6aR)-2-cyclopentyl-5-(1,3-thiazol-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}piperidine-4-carboxamide
N-{2-methyl-3-[({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)carbamoyl]phenyl}oxolane-2-carboxamide
N-[2-(ethanesulfonyl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
4-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)thiomorpholine
6-(morpholin-4-yl)-N-[(4-phenyloxan-4-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
14-(2-tert-butylpyrimidin-5-yl)-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
1-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}-4-ethyl-1,4-diazepane
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(5-fluoropyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(6-fluoro-1H-1,3-benzodiazole-2-carbonyl)-1,4-diazepane-6-carboxylic acid
4-({[2-(2-methoxyphenoxy)ethyl]amino}methyl)benzene-1-sulfonamide
1-ethyl-5-[methyl({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl})amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-methoxy-1-{1'-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
3-{[1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl}benzoic acid
N,N-dimethyl-1-{[2-(1H-1,2,4-triazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]sulfonyl}pyrrolidin-3-amine
5-chloro-7-methoxy-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-benzofuran-2-carboxamide
2-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-1-carbonyl)-1H-indole
3-{[4-(4-methoxyphenoxymethyl)piperidin-1-yl]methyl}piperidin-3-ol
1-{5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}-5-phenylpentane-1,5-dione
3-(2-{[1-(1,3-benzothiazol-2-yl)piperidin-4-yl]amino}ethyl)-1,3-oxazinan-2-one
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3-(2-ethyl-1H-1,3-benzodiazol-1-yl)propanamide
5-{[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1,3-oxazolidin-2-one
(2R,6R)-6-methyl-1-[(4-methyl-1H-imidazol-5-yl)methyl]-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
2-(2-ethyl-1H-imidazol-1-yl)-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}acetamide
(2S,4R)-4-(4-cyanobenzamido)-N-ethyl-1-(pyridin-2-ylmethyl)pyrrolidine-2-carboxamide
4-(4-{pyrazolo[1,5-a]pyridine-7-carbonyl}piperazin-1-yl)quinazoline
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
3-[6-(2-methoxyphenyl)pyridazin-3-yl]-7-methyl-1H-indole
N-(1-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
3-[ethyl({[2-(furan-2-yl)pyrimidin-5-yl]methyl})amino]-1λ6-thiolane-1,1-dione
8-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
6-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
N,1-dimethyl-N-[2-(morpholin-4-yl)propyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 2-[(butan-2-yl)sulfamoyl]-6-(2-chloro-4-fluorobenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-methyl-3-(pyrrolidin-1-yl)propan-1-one
5-cyclopropyl-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
N-(2-chloro-5-methylphenyl)-6-(hydroxymethyl)-1,4-oxazepane-4-carboxamide
2-butyl-8-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
3-(oxolan-3-yl)-1-{4-[(trifluoromethyl)sulfanyl]phenyl}urea