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2-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-phenyl-N-[(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-3-yl)methyl]methanesulfonamide
2-{[(1-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
(3S,5S)-1-[(3-fluoro-2-methylphenyl)methyl]-5-[(4-fluorophenyl)carbamoyl]piperidine-3-carboxylic acid
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-decahydro-1,6-naphthyridin-2-one
2-(2,1,3-benzoxadiazol-4-ylmethyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
2-(2-hydroxyethyl)-9-(2-methylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-(6-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-2-yl)ethan-1-ol
4-[({[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)methyl]-1-ethylpyrrolidin-2-one
N-[(4-fluorophenyl)methyl]-N-methyl-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
1-ethyl-5-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-{[6-(morpholin-4-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}furan-3-carboxamide
4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-methyl-1-[(4-methylphenyl)methyl]piperazin-2-one
N-methyl-2-(methylsulfanyl)-N-[(1-phenylpyrrolidin-3-yl)methyl]benzamide
5-[4-(morpholin-4-yl)piperidine-1-carbonyl]-N-propylpyridin-2-amine
1-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
1-(1H-imidazol-1-ylmethyl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}cyclopropane-1-carboxamide
1-(4-{[2-(dimethylamino)ethyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
5-chloro-2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)phenol
[2-(azepan-1-yl)ethyl](ethyl){[4-(pyrimidin-5-yl)phenyl]methyl}amine
2-{2-[(1R,3R,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]-2-oxoethyl}-4-phenyl-1,2-dihydrophthalazin-1-one
(4aS,7aR)-1-(1H-imidazol-4-ylmethyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[1-(2-propyl-1,3-thiazole-4-carbonyl)azetidin-3-yl]pyridine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(furan-3-ylmethyl)piperidin-3-ol
4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]thiomorpholine
4-{[5-(2,3-dichlorophenyl)furan-2-yl]methyl}-2-(trifluoromethyl)morpholine
2-methyl-6-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-2,3-dihydropyridazin-3-one
2-(1-{[1-(1,3-benzothiazole-2-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
[(3R,4R)-1-(2-amino-6-methylpyrimidin-4-yl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
[(3S,5R)-1-[(3,5-difluoro-4-methoxyphenyl)methyl]-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
N-(5-methyl-1,2-oxazol-3-yl)-2-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoacetamide
N-[2-(2-chlorophenyl)ethyl]-3-(pyrrolidin-3-yl)benzamide
4-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-2,6-dimethylpyrimidine
1-(2-amino-6-methoxypyrimidin-4-yl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2,2,2-trifluoroethyl)propanamide
2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)acetamide
N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]cyclohexanecarboxamide
4-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1,2-dihydroquinolin-2-one
N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
3-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
8-(2-methyl-1-benzofuran-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[3-(methylsulfanyl)propyl]benzamide
(3R,5R)-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
4-[4-(2-ethylbutyl)piperazin-1-yl]-2-[(2-fluorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
(2R,3R,6R)-3-(4-fluorophenyl)-5-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[3-(cyclopropylcarbamoyl)-5-{[(5-ethylfuran-2-yl)methyl]amino}benzenesulfonyl]piperidine-3-carboxamide
1-[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]-2-methyl-1,4-diazepan-5-one
N-[3-(pyridin-2-yl)propyl]-6-{[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]amino}pyridine-3-carboxamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-[1-(pyrimidin-4-yl)ethyl]propanamide
2-methyl-6-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}pyridine