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(4aS,7aR)-1-[(4-methylphenyl)methyl]-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{4-[4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}-2,3-dihydro-1H-inden-1-one
8-chloro-2-(furan-2-yl)-N-(oxan-3-ylmethyl)quinoline-4-carboxamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-[2-(furan-2-yl)phenyl]-1H-imidazole
3-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(dimethylamino)-N-(2-methoxyethyl)-4-methyl-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
1-(3-methoxyphenyl)-4-(3-propoxypiperidin-1-yl)piperidine
3-(4-hydroxyphenyl)-N-(2-methoxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrazole-5-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{2H,3H-thieno[3,4-b][1,4]dioxin-5-ylformamido}acetic acid
2-(4-fluorophenyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridine
{4-methyl-5-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methanol
2-cyclopropanecarbonyl-8-[3-(1H-pyrazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1H-pyrrole-2-carbonyl)-1,4-diazepan-6-ol
N-ethyl-2-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
5-(2-fluorophenoxymethyl)-N-(1H-1,2,4-triazol-3-ylmethyl)-1H-pyrazole-3-carboxamide
1-[4-(furan-2-yl)pyrimidin-2-yl]-N-[(2-methoxyphenyl)methyl]-5-methyl-1H-pyrazole-4-carboxamide
4-(5-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
(3S,4R)-1-[2-(2-hydroxyethoxy)ethyl]-4-phenylpyrrolidine-3-carboxylic acid
1-(1H-imidazol-2-ylmethyl)-4-phenoxypiperidine-4-carboxylic acid
(5R)-5-[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
6-{[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
2-[(1-methylpiperidin-4-yl)methyl]-2,8-diazaspiro[4.5]decane
2-(2-methyl-1H-imidazol-1-yl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}propanamide
5-(azocan-1-yl)-1-methyl-N-[2-(piperidin-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-{[2-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-1H-imidazol-1-yl]methyl}-1,2-oxazole
{3-[(2,4-difluorophenyl)methyl]-1-(quinoxalin-2-yl)piperidin-3-yl}methanol
2-(cyclopropylmethyl)-8-{2-[4-(dimethylamino)phenyl]acetyl}-2,8-diazaspiro[5.5]undecan-3-one
1-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]-4-phenylpiperazine
4-[4-(3-methylpyridin-4-yl)piperazine-1-carbonyl]-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-[2-(5-methylfuran-2-yl)propyl]-1H-1,2,3-triazole
(3S,7S,8aS)-3-(4-aminobutyl)-7-{[(2-fluorophenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
8-(5-carboxypyridin-2-yl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H-imidazol-2-yl)pyridine
1-[(4-methoxyphenyl)methyl]-4-(piperidin-3-ylmethyl)piperazin-2-one
5-ethyl-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-[4-(4-benzylpiperazine-1-carbonyl)-5-cyclopropyl-1H-pyrazol-1-yl]-4-(5-methylfuran-2-yl)pyrimidine
1-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}-N,4-dimethylpiperidine-4-carboxamide
3,4-dichloro-N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]benzamide
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]benzamide
5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-N-(pyridin-2-ylmethyl)pyridin-2-amine
(3S,4R)-N,N-dimethyl-1-(naphthalene-2-carbonyl)-4-(propan-2-yl)pyrrolidin-3-amine
(4-{5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}phenyl)methanol
{2-[6-(4-fluorophenyl)pyridazin-3-yl]phenyl}methanol
3-(1H-1,2,3-benzotriazol-1-yl)-1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]propan-1-one
1-methyl-3-(1-oxo-2,3-dihydro-1H-inden-5-yl)-1-[1-(pyridin-3-yl)pentyl]urea
N-[2-(dimethylamino)pentyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
8-(dimethyl-1,3-oxazole-5-carbonyl)-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(pyridin-2-yl)propanamide
3-(pentan-2-yl)-8-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2-methoxyethyl)-2-(pyridin-2-ylsulfanyl)-N-(thiophen-2-ylmethyl)propanamide