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({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[3-(3-phenylpropanoyl)piperidin-1-yl]acetamide
3-{[(2,2-dimethyloxan-4-yl)amino]methyl}-7-methyl-1-(2-phenoxyethyl)-1,2-dihydroquinolin-2-one
N-(adamantan-2-ylmethyl)-2-ethyl-6-methyl-4-oxo-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl){[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}amine
3,5-dimethyl-1-[(4-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}phenyl)methyl]-1H-pyrazole
(3aR,7aS)-2-(2-ethylpyrimidine-5-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
(3aS,6aS)-2-methanesulfonyl-5-(2-phenoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-cyclopropyl-1-[1-(thiophen-3-yl)propan-2-yl]-1H-imidazole
5-[(4-benzylpiperidin-1-yl)methyl]-N-[(2S)-1-hydroxy-3-methylbutan-2-yl]-1,2-oxazole-3-carboxamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(1H-pyrazol-1-yl)benzamide
3-methyl-8-(4-methyl-3,4-dihydro-2H-1,4-benzoxazine-7-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-cyclopropyl-N-(2-phenyl-1-{1-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]piperidin-4-yl}ethyl)pyridine-2-carboxamide
2-chloro-4-[1-(3,4-dimethoxyphenyl)-1H-imidazol-2-yl]phenol
N4-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-5,6-dimethylpyrimidine-2,4-diamine
4-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyrrolidin-2-one
(4aS,8aR)-6-(5-ethylpyrimidin-2-yl)-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
4-ethyl-3-(2-oxo-2-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethyl)piperazin-2-one
3-(3-fluorophenyl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]propan-1-one
1-(propan-2-yl)-4-{1-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-1H-imidazol-2-yl}piperidine
N4-[(3,4-dimethoxyphenyl)methyl]-5-ethylpyrimidine-2,4-diamine
N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-5-propyl-1,3,4-oxadiazol-2-amine
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
7-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
1-(thiophen-2-ylmethyl)-4-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]piperazine
2-{2-[(2,2-dimethylmorpholin-4-yl)methyl]-6-methoxyphenoxy}propanoic acid
(2S,4S)-N-ethyl-1-(propan-2-yl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
4-[3-(oxan-4-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]cyclohexan-1-ol
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylpropyl)acetamide
5-{1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}-3-methyl-1,2-oxazole
2-(ethylamino)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]pyrimidine-5-carboxamide
2-(1-methylpiperidin-4-yl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
(3R)-N-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-amine
3-(3-fluorophenyl)-4-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
2-(propan-2-ylsulfanyl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
{3-propyl-1-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperidin-3-yl}methanol
(3aS,6aS)-2-cyclohexyl-5-({3-[(dimethylamino)methyl]phenyl}methyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-ethyl-4-phenyl-9-(pyridine-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-3-methylbut-2-en-1-one
N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
6-cyclopentyl-N,1-dimethyl-N-[(3-methylpyridin-2-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(cyclopentylmethyl)-6-methyl-4-oxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
3-{1-[benzyl(methyl)sulfamoyl]piperidin-3-yl}benzoic acid
1-{6-methyl-3-[(4-methylpiperazin-1-yl)methyl]quinolin-2-yl}piperidin-3-ol
N-(1-{[5-(4-ethoxyphenyl)furan-2-yl]methyl}piperidin-3-yl)acetamide
5-ethyl-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)pyrimidin-2-amine
4-[(benzyloxy)methyl]-1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}thiophene-3-carboxamide
2-(3-hydroxypiperidin-1-yl)-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]acetamide
3-(4-methoxy-3,5-dimethylbenzoyl)-1-(thian-4-yl)piperidine