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5-{[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]methyl}-N-methylfuran-2-carboxamide
3-(3-fluorophenyl)-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
2-({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}amino)-N-(1,3-thiazol-2-yl)propanamide
2-[1-(5-chloro-2-methoxyphenyl)-5-[(R)-cyclohexyl(hydroxy)methyl]-1H-1,2,4-triazol-3-yl]acetamide
N-[(3-methylphenyl)methyl]-N-(propan-2-yl)-2-(pyridin-2-yl)pyrimidine-5-carboxamide
1-acetyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]piperidine-4-carboxamide
5-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-3-(2-phenylethyl)-1H-1,2,4-triazole
1-(1-{[2-methyl-5-(1,2-oxazol-5-yl)furan-3-yl]sulfonyl}piperidin-3-yl)pyrrolidin-2-one
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amino]acetamide
N3-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-N5-(2,2,2-trifluoroethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(2,3-dihydro-1H-inden-2-yl)-2,5,7-trimethyl-N-propylpyrazolo[1,5-a]pyrimidine-3-carboxamide
5-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridine-2-carbonitrile
4-(2-methoxypyridine-4-carbonyl)-3-methyl-1-[(3-methylphenyl)methyl]piperazin-2-one
dimethyl({4-[1-(1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]phenyl}methyl)amine
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[2-(3-phenoxyphenyl)ethyl]acetamide
N4-cyclopentyl-7-(oxolane-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
(3R,5R)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
3-[(5-ethylpyridin-2-yl)methyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
1-{[3-cyclopropyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-(2-{[6-methyl-2-(morpholin-4-yl)pyrimidin-4-yl]amino}ethyl)piperidin-3-ol
3-hydroxy-1-(2-methoxyethyl)-3-{[(pyridin-4-ylmethyl)amino]methyl}piperidin-2-one
1-methyl-3-(3-methyl-1-propyl-1H-pyrazol-5-yl)-1-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}urea
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-methyl-3-[5-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]urea
8-[(2-methoxyphenyl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}pyrrolidin-3-yl]acetamide
1-methyl-9-(prop-2-en-1-yl)-4-(pyrrolidine-1-sulfonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(furan-2-ylmethyl)-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}piperidine-4-carboxamide
N-(4-{1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-imidazol-2-yl}phenyl)acetamide
2-{[3-(1-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
6-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-2-(2-hydroxyethyl)-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
1-(3-methoxyphenyl)-4-[(6-methylquinolin-5-yl)methyl]piperazin-2-one
(3S,4R)-1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-4-(3-methylthiophen-2-yl)piperidin-3-ol
5-(2-methyl-4-phenylpiperazine-1-carbonyl)pyrazin-2-ol
4-{1-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1H-imidazol-2-yl}pyridine
3-{[(cyclohex-1-en-1-ylmethyl)carbamoyl]amino}-4-methoxy-N-methylbenzamide
2,7-dimethyl-N-[2-(pyrrolidin-1-yl)ethyl]quinoline-4-carboxamide
N-benzyl-N-(3-hydroxy-2-methylpropyl)-2-(phenylformamido)acetamide
N-{1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]pyrrolidin-3-yl}acetamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(3,4-dimethoxybenzoyl)piperidine-3-carboxylate
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-4-(2-oxopiperidin-1-yl)butanamide
(2R,6R)-4-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-amine
1-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2-(2,3-dihydro-1H-inden-1-yl)ethan-1-one
N-{1-[(cyclopropylcarbamoyl)methyl]piperidin-4-yl}-3-(1H-imidazol-2-yl)benzamide
2-(5-{[3-chloro-2-oxo-5-(trifluoromethyl)-1,2-dihydropyridin-1-yl]methyl}-3-methyl-1H-1,2,4-triazol-1-yl)acetic acid
(3R,5S)-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
8-[2-(propan-2-ylsulfanyl)ethyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(2,3-difluoro-4-methoxybenzoyl)-3-(3-methoxypropyl)piperidine
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide