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N-[(4-fluorophenyl)methyl]-2,3,4-trimethoxy-N-(prop-2-en-1-yl)benzamide
2-[6-(4-chloro-3-fluorophenyl)pyridin-3-yl]acetic acid
2-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}acetic acid
4-({4-[6-oxo-4-(oxolan-2-yl)-1,6-dihydropyrimidin-2-yl]phenyl}methyl)-1,4-diazepan-2-one
{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}[(2-methoxyphenyl)methyl]amine
1-[2-(1H-imidazol-2-yl)benzoyl]-4-(piperidine-1-carbonyl)piperidine
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl]propan-1-ol
4-{[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}benzonitrile
1-(azepan-2-ylmethyl)-3-[3-(2-ethoxyethoxy)phenyl]urea
4-tert-butyl-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
7-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-2-oxa-7-azaspiro[4.5]decane
methyl({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)(oxan-2-ylmethyl)amine
3-(1H-imidazol-1-ylmethyl)-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidine
N-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-ethylbenzamide
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1-methyl-1H-pyrazol-4-yl)propanamide
(1R,5R)-6-[3-(methylsulfanyl)propyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3R,5S)-N3-[(3-fluoro-4-methylphenyl)methyl]-N5-(4-methylphenyl)piperidine-3,5-dicarboxamide
4-[4-(1-cyclopentylpiperidine-3-carbonyl)piperazin-1-yl]-5,6-dimethylpyrimidine
N-cyclopropyl-4-methyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)benzamide
1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
N-(1-methyl-1H-1,2,3-triazol-4-yl)-3-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}benzamide
N-(5-methyl-1,2-oxazol-3-yl)-4-oxo-3,4-dihydrophthalazine-1-carboxamide
(4aR,7aS)-1-(1H-imidazol-2-ylmethyl)-4-{[1-(propan-2-yl)piperidin-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3,6-dimethyl-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-benzofuran-2-carboxamide
2-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}imidazo[1,2-a]pyrimidine-3-carboxamide
2-(adamantan-1-yl)-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methylacetamide
ethyl 4-(2-phenoxyethyl)-1-(1,3-thiazole-5-carbonyl)piperidine-4-carboxylate
3-[({1-[(2,3,4-trifluorophenyl)methyl]piperidin-3-yl}oxy)methyl]pyridine
2-[3-(1H-imidazol-1-yl)propyl]-9-[3-(methylsulfanyl)butyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-benzyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
2-methoxy-1-[1'-(4-methyl-1H-imidazole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
3-(1-{3-azaspiro[5.5]undecan-9-yl}piperidin-4-yl)phenol
1-methyl-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
4-[1-(3-fluoro-4-methoxybenzoyl)piperidin-4-yl]-5-phenyl-2-(pyridin-3-yl)pyrimidine
9-(1-benzyl-1H-pyrazole-4-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
6-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-chloro-N-{1-phenyl-3,6-diazatricyclo[4.3.1.13,8]undecan-9-yl}furan-2-carboxamide
1-benzyl-N3-cyclopentyl-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
3-({[2-(1H-imidazol-1-yl)ethyl](methyl)amino}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
(3S,5S)-1-methyl-5-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrrolidin-3-amine
2-[4-({[2-(1H-imidazol-1-yl)ethyl](methyl)amino}methyl)phenoxy]-1-(morpholin-4-yl)ethan-1-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(3-hydroxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-butyl-N-methyl-3-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
N-[2-(furan-2-yl)ethyl]-7-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
6-chloro-2-{[4-(1H-pyrazol-3-yl)piperidin-1-yl]methyl}quinolin-4-ol
5-methyl-4-(3-methyl-1H-pyrazole-5-carbonyl)-1-(3-phenylphenyl)piperazin-2-one
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-(pyridin-3-yl)acetamide
N-cyclopropyl-3-[5-(5-ethyl-2-methylpyrimidin-4-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
3-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide