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N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
1-[1-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
2-cyclohexyl-N-(3-ethoxy-2-hydroxypropyl)-1,3-benzoxazole-6-carboxamide
5-{[(3-methoxyphenyl)methyl](methyl)amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-({[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amino}methyl)benzoic acid
N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)-1H-pyrazole-3-carboxamide
(1-methyl-1H-imidazol-2-yl)[1-(6-methylquinoline-4-carbonyl)piperidin-4-yl]methanol
[(3-{2-[4-(2,3-dimethyl-1H-indole-7-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(1,3-thiazol-4-ylmethyl)amine
4-[2-(3,4-dichlorophenyl)morpholin-4-yl]butanoic acid
2-(azepan-1-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidine
1-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]-4-(pyridin-2-yl)piperidin-4-ol
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-acetyl-N-[(5-methylpyrazin-2-yl)methyl]thiophene-3-carboxamide
2-{4-[3-(4-benzylpiperidin-1-yl)-3-oxopropyl]piperidin-1-yl}-2-oxoacetamide
N-[2-(ethylsulfanyl)ethyl]-2-(pyrrolidin-3-yl)benzamide
1-{1'-[2-(1H-imidazol-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
7-(3,6-dimethylpyrazin-2-yl)-4-(3-methylfuran-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-[1-(2-ethylpyrimidine-5-carbonyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
(1R,3S)-3-(2-aminoethoxy)-7-(5-methylpyridine-3-carbonyl)-7-azaspiro[3.5]nonan-1-ol
(isoquinolin-5-ylmethyl)[2-(4-methoxyphenoxy)ethyl]methylamine
2-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidine-1-carbonyl}-1,4-dihydroquinolin-4-one
N-tert-butyl-3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}urea
1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
(2S,4S)-4-amino-N,N-diethyl-1-[(1-ethyl-1H-pyrazol-5-yl)sulfonyl]pyrrolidine-2-carboxamide
3-[5-(4-fluoro-2-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]-1λ6-thiolane-1,1-dione
N,N-diethyl-1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperidine-3-carboxamide
2-methyl-6-{1-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1H-imidazol-2-yl}pyridine
N-(2H-1,3-benzodioxol-5-yl)-2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
2-(4-methoxyphenyl)-N-({1-[(2-methyl-1H-indol-3-yl)methyl]piperidin-3-yl}methyl)acetamide
ethyl 1-{imidazo[2,1-b][1,3]thiazole-6-amido}cyclobutane-1-carboxylate
4,4,4-trifluoro-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}butan-1-one
1-(1H-imidazol-4-ylmethyl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
(2S,4S)-N-ethyl-1-{[3-(furan-2-yl)phenyl]methyl}-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
2-(4-fluoro-2-methoxyphenyl)-2-[4-(morpholin-4-ylmethyl)piperidin-1-yl]acetic acid
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-(2-oxopiperidin-1-yl)acetamide
2-[3-(2-phenylethyl)-5-(pyridin-3-ylmethyl)-1H-1,2,4-triazol-1-yl]pyridine
1-[2-methyl-5-(4-methyl-2-phenylpiperazine-1-carbonyl)phenyl]imidazolidin-2-one
(1R,5R)-3-{[5-(dimethyl-1,2-oxazol-5-yl)furan-2-yl]sulfonyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonane
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(5-methylfuran-2-yl)benzamide
(3R,4S)-4-cyclopropyl-1-(4-fluorobenzoyl)-N,N-dimethylpyrrolidin-3-amine
N3-butyl-1-(furan-2-ylmethyl)-N5-[(2-methylphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-cyclopropyl-N-{2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-5-carboxamide
5-(3-methoxyphenoxymethyl)-N-[2-(1H-pyrazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
2-amino-6-(4-hydroxyphenyl)-5-methyl-4-{2-[(propan-2-yl)amino]pyrimidin-5-yl}pyridine-3-carbonitrile
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}piperidin-2-one
2-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidine-1-carbonyl]pyridin-3-ol
4-benzyl-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}pyrrolidin-2-one
3-fluoro-2-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine