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(1S,4S)-5-(2-aminoacetyl)-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
3-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-2,2-dimethylpropan-1-ol
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-6-phenyl-5,6,7,8-tetrahydroquinoline-3-carbonitrile
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}furan-2-carboxamide
2-ethyl-8-[(3-methylphenyl)methanesulfonyl]-2,8-diazaspiro[5.5]undecan-3-one
(2R,6R)-11-methoxy-4-(1,3-thiazol-2-ylmethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-(pyridin-2-ylmethyl)-1-[1-(pyridine-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
ethyl 3-({3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}amino)propanoate
4-(3-hydroxy-3-methylbutyl)-N-[1-(methoxymethyl)cyclopentyl]benzamide
(1R,2R,4R)-N-({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
N-({7-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)propane-2-sulfonamide
7-[3-(1H-indol-1-yl)propyl]-2-oxa-7-azaspiro[4.5]decan-8-one
6-(4-chlorophenyl)-N-[(2S)-1-hydroxybutan-2-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
methyl 2-{1-[3-(1,2-oxazinan-2-yl)propanoyl]-3-oxopiperazin-2-yl}acetate
2-(2-fluoro-5-methoxyphenyl)-1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazole
5-(3-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propyl)-1,3,4-thiadiazol-2-amine
2-(3-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}phenoxymethyl)pyridine
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-{3-[(3-chloro-4-fluorophenyl)carbamoyl]propanamido}propanoic acid
2-(cyclopent-1-ene-1-carbonyl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
2-(2-ethoxynaphthalen-1-yl)-N,N-dimethylpyridine-3-carboxamide
1-[1-(4-methylpentanoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
8-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2,4-dimethyl-6-[3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carbonitrile
2-(2-methylbutyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{3-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidine-1-carbonyl]phenyl}ethan-1-one
2-ethoxy-1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
4-{4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine-1-carbonyl}imidazolidin-2-one
5-acetyl-N-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(3S,4R)-4-(pyridin-3-yl)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidine-3-carboxylic acid
8-cyclopropanecarbonyl-2-[2-(2,5-dimethylphenyl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(1S,4R)-2-{[1-(4-methylpyridin-2-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]methyl}-2-azabicyclo[2.2.1]heptane
4-{[1-(2-phenylpropyl)piperidin-4-yl]oxy}-N-(pyridin-4-ylmethyl)benzamide
N-(2,3-dihydro-1H-inden-2-yl)-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
N-methyl-2-{3-oxo-2-azaspiro[4.4]nonan-2-yl}-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
N-({1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)-1H-pyrrole-2-carboxamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)thiophene-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-(2-ethylpiperidine-1-carbonyl)-5-methylthieno[2,3-d]pyrimidin-4-amine
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-(furan-2-ylmethyl)-N-methyl-1H-pyrazole-4-carboxamide
1-methyl-1-[(5-methylfuran-2-yl)methyl]-3-[5-(4-methylphenyl)-1,3,4-thiadiazol-2-yl]urea
[(2S,6S)-4-[(1-ethyl-1H-indol-4-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
8-{6-[(propan-2-yl)amino]pyrimidin-4-yl}-2,8-diazaspiro[4.5]decan-3-one
2-[4-(hydroxymethyl)phenyl]-2-{methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}acetic acid
2-{3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl}phenol
(1R,5S,8R)-3-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-3-azabicyclo[3.2.1]octan-8-ol
N-cycloheptyl-3-(2-phenylethyl)-1H-1,2,4-triazole-5-carboxamide
3-{[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]methyl}pyrrolidin-3-ol
9-(4-aminopyrimidin-2-yl)-2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-{2-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
6-(3,4-dimethylpiperazin-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide