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2-[1-(4,6-dimethylpyrimidin-2-yl)-1H-pyrazol-4-yl]-N,N,8-trimethylquinoline-4-carboxamide
7-{[2-(methoxymethyl)piperidin-1-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-(butan-2-yl)-7-[(2H-1,2,3,4-tetrazol-5-yl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
4-(3-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}phenyl)-2-methylbut-3-yn-2-ol
N3-cyclohexyl-N5-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
8-[2-(methylamino)pyridine-4-carbonyl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
1-(2-ethoxyphenyl)-2-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(3-fluorophenyl)-1,3-benzoxazole-5-carboxamide
{5-[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methanol
4-(1,3-benzoxazol-2-yl)-N-(dimethyl-1,2-oxazol-4-yl)piperidine-1-carboxamide
5-[({[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)methyl]pyrimidin-2-amine
4-ethyl-3-{1-[3-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[4-(ethylcarbamoyl)-2-methylphenyl]-2-(morpholin-4-ylmethyl)piperidine-1-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-5-hydroxypyrazine-2-carboxamide
2-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[(3aR,6aR)-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-4-(4-methoxyphenoxymethyl)piperidine
N-[3-(pyridin-4-yl)propyl]-6-[3-(trifluoromethyl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[1-(4-methoxyphenyl)-3-methyl-1H-pyrazol-5-yl]-3-[3-(methylsulfanyl)propyl]urea
[(2-chloropyridin-3-yl)methyl](methyl){[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amine
1-benzyl-8-(2,2-diphenylethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-1-[3-(methylsulfanyl)butyl]piperidine
7-[(3,4-difluorophenyl)methyl]-2-(4-methylpentanoyl)-2,7-diazaspiro[4.5]decan-6-one
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}benzamide
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-2-methylfuran-3-carboxamide
(4aS,7aR)-1-(2,5-dimethylfuran-3-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-N-(3-methylphenyl)methanesulfonamide
2-[5-(5-phenyl-1H-pyrazole-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
N-[(2-ethoxypyridin-3-yl)methyl]-2,3-dimethylquinoxaline-6-carboxamide
4-[(2-{1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
3-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
(3R,5S)-N-[2-(1H-imidazol-4-yl)ethyl]-1-(2-methylpropyl)-5-[(pyridin-3-yloxy)methyl]piperidine-3-carboxamide
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-ethoxyphenyl)ethan-1-one
N,2,6-trimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]quinoline-4-carboxamide
2-{1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
dimethyl[(4-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-2-yl}phenyl)methyl]amine
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N,5-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
3-(hydroxymethyl)-1-(2-methyl-4-phenylpyrimidine-5-carbonyl)piperidin-3-ol
N-({1-[(3-methyl-1H-indol-2-yl)methyl]pyrrolidin-3-yl}methyl)pyrazine-2-carboxamide
3-hydroxy-1-(2-phenylethyl)-3-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-ylmethyl}piperidin-2-one
3-[2-(dimethylamino)ethyl]-1-[2-fluoro-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-(oxolan-2-ylmethyl)urea
2-[3-(3-methylbutyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl]pyrrolidine-1-carboxamide
1,6-dimethyl-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-cyclohexyl-N-[1-(pyrazin-2-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
N-phenyl-3-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}propanamide
2-(dimethylamino)-N-(furan-2-ylmethyl)-N-methyl-2-(3-methylphenyl)acetamide
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[(2,6-difluorophenyl)methyl]pyrrolidin-2-one
2-amino-6-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-4-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-(8-chloro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}urea
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1,1-dioxo-1λ6-thiane-4-carboxamide
5-[3-(aminomethyl)pyrrolidine-1-carbonyl]-2-[(2,6-dichlorophenyl)methyl]pyrimidin-4-ol