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(4aR,7aS)-1-ethyl-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2R)-2-({[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}amino)propanamide
8-[2-(morpholin-4-yl)acetyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
7-(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
7-chloro-3,5-dimethyl-N-{3-[(pyridin-3-yl)amino]propyl}-1-benzofuran-2-carboxamide
3-[5-({7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)thiophen-2-yl]prop-2-yn-1-ol
N-[(5-methylpyrazin-2-yl)methyl]-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanamide
1-(3-phenylpropyl)-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]piperidin-2-one
N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyacetyl)pyrrolidin-3-yl]-4-(propan-2-yl)-1,3-thiazole-2-carboxamide
4-chloro-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-1-methyl-1H-pyrazole-5-carboxamide
2-fluoro-N-methyl-5-({[(1R,2S)-2-phenylcyclohexyl]carbamoyl}amino)benzamide
5-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-1H-1,3-benzodiazole
4-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-2-(trifluoromethyl)morpholine
1-(2-{1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
2-{[1-(2-fluorophenyl)cyclopentyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
(3R,9aR)-3-methyl-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{[5-(4-fluorophenyl)furan-2-yl]methyl}-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
8-(2-methylquinolin-4-yl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]-1,8-diazaspiro[4.5]decane
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
2-(dimethylamino)-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(4-fluorophenyl)ethan-1-one
1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-methyl-3-[5-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]urea
8-(4-acetyl-6-hydroxy-1,4-diazepane-1-carbonyl)-2-methyl-1,4-dihydroquinolin-4-one
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(2-phenoxyethyl)piperazine
3-{1-[2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
N-methyl-1-(2-phenylethyl)-5-[4-(piperidin-1-yl)piperidin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-(2,6-dimethylpyridine-4-carbonyl)-N,N-dimethylpiperazine-1-carboxamide
2-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]-1H-imidazol-2-yl}-1H-1,3-benzodiazole
2-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-5-methoxy-4H-pyran-4-one
1-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]-3-(3-methoxyphenoxymethyl)piperidine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-methanesulfonyl-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamido)-1H-indole-3-carboxamide
N-benzyl-2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
5-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-(2,3-dihydro-1H-inden-2-yl)-N-[3-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
2-(adamantan-1-yl)-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]acetamide
1-({2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}methyl)-4-hydroxypiperidine-4-carboxylic acid
2-[1-(4-methoxyphenyl)-5-(morpholin-2-ylmethyl)-1H-1,2,4-triazol-3-yl]acetamide
2-[2-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]-4,6-dimethylpyridine-3-carbonitrile
(4aR,7aS)-1-(cyclopropylmethyl)-4-[3-(4-methoxyphenyl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperidin-4-ol
4-(1-methyl-1H-imidazol-2-yl)-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidine
4-{1-[(5-methylthiophen-2-yl)sulfonyl]azetidin-3-yl}pyridine
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(oxan-4-yl)acetamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
4-[(2S)-1-{[2-(cyclopentyloxy)phenyl]methyl}pyrrolidine-2-carbonyl]morpholine
7-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
7-(cyclohexylmethyl)-2-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]cyclopropane-1-carboxamide
3-fluoro-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide