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5-{1-[(5-chlorofuran-2-yl)methyl]pyrrolidin-2-yl}-3-methyl-1H-1,2,4-triazole
2-amino-4-[1-(4-methoxyphenyl)-1H-pyrrol-2-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-ethyl-9-[(4-methyl-1H-imidazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
7-propyl-2-(quinoxalin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
5-methyl-N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)pyrazine-2-carboxamide
[(3R,5R)-1-(2-methoxypyridine-4-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
2-(adamantan-1-yl)-N-{1-azabicyclo[2.2.2]octan-3-yl}acetamide
2-ethyl-5-{4-[4-(4-methylphenyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}pyrimidine
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl){[5-(oxolan-2-yl)thiophen-2-yl]methyl}amine
4-{[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]amino}-1-propylpyrrolidin-2-one
1-methyl-4-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
1-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-N-(2,3-dihydro-1,4-benzodioxin-6-yl)piperidin-3-amine
methyl (2S)-2-({5-[(2-methylpropyl)carbamoyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridin-3-yl}formamido)-2-phenylacetate
2-[3-({[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2-methyl-1H-indol-1-yl]acetamide
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-5-phenyl-1,2-oxazole-4-carboxamide
N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
N-(3-cyanophenyl)-2-(3-methoxypropyl)piperidine-1-carboxamide
1-(4-phenylbutan-2-yl)-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
(3R)-N-(3-chloro-2-propoxyphenyl)-3-hydroxypyrrolidine-1-carboxamide
(2S,4S)-4-amino-N,1-dimethyl-N-{[3-(methylsulfanyl)phenyl]methyl}pyrrolidine-2-carboxamide
1-(4,6-dimethylpyrimidin-2-yl)-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]piperidin-4-amine
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(3-methoxypyrazin-2-yl)pyrrolidin-3-yl]methanol
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-(2-hydroxyethyl)-N-propylpropanamide
1-(2-chlorophenyl)-3-(1-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(4-methyl-1,3-thiazol-5-yl)methyl]piperidine
7-(9H-fluorene-9-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}({[3-(trifluoromethoxy)phenyl]methyl})amine
2-(dimethylamino)-2-(3-fluorophenyl)-N-methyl-N-(quinolin-2-ylmethyl)acetamide
4-ethyl-3-[(1-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-oxo-2H-chromene-3-carboxamide
2-[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole
2-[3-(2-methoxyethyl)-5-(5-methoxyfuran-2-yl)-1H-1,2,4-triazol-1-yl]benzoic acid
N-[(5-methylpyrazin-2-yl)methyl]-3-(piperidin-4-ylmethyl)benzamide
1-[1-(1H-indol-5-yl)ethyl]-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{2-[4-(propan-2-yloxy)phenyl]ethyl}acetamide
3-cyclopentyl-1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
4-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-1-methylpiperazine-2-carboxylic acid
N-(3-phenylprop-2-yn-1-yl)-N-propylimidazo[1,2-a]pyridine-6-carboxamide
14-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(pyridin-4-ylmethyl)piperidin-3-amine
N-cyclopentyl-N-[(5-methylthiophen-2-yl)methyl]-2-(pyridin-3-yloxy)acetamide
(1R,5S,6S)-6-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-3-azabicyclo[3.1.0]hexane
4-[(1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidin-2-yl)methyl]morpholine
[(3S,5R)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(1,3-thiazole-4-carbonyl)piperidin-3-yl]methanol
N-(2-chloro-6-methylphenyl)-6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decane-2-carboxamide
5-[2-(dimethylamino)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
5-tert-butyl-4-[(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)methyl]furan-2-carboxamide