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N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-5-chloro-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-methyl-4-(2,3,4-trimethoxyphenyl)-1H-pyrazol-5-amine
1-(2-chlorophenyl)-3-{1-[1-(4-methylpentan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
(2S,4R)-N-ethyl-4-(3-fluoro-4-methylbenzamido)-1-(furan-3-ylmethyl)pyrrolidine-2-carboxamide
4-(1-cyclopropyl-6-oxopiperidine-3-carbonyl)-1-phenylpiperazin-2-one
1-(1,3-dihydro-2-benzofuran-5-yl)-3-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]urea
3-(3-hydroxy-3-methylbutyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]benzamide
1-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidin-4-amine
7-(cyclopropylmethyl)-2-[2-(2,3-dimethylphenoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one
3-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-(2-chloropyridin-3-yl)urea
N-[3-(dimethylamino)propyl]-1-[(2-fluoro-4-methoxyphenyl)methyl]-N-methylpiperidin-3-amine
1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-4-(morpholin-4-yl)butan-1-one
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[4-(2-propoxyethyl)piperazin-1-yl]ethan-1-one
N-[(4-fluorophenyl)methyl]-3-(2-hydroxyphenyl)-N-(3-hydroxypropyl)-1H-pyrazole-5-carboxamide
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-6-(methoxymethyl)pyridine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-1-phenylcyclopropane-1-carboxamide
N-(2,5-difluorophenyl)-2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide
2-amino-4-(2-butyl-1H-imidazol-4-yl)-6-(2-hydroxypropan-2-yl)pyridine-3-carbonitrile
1-{1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-4-yl}pyrrolidin-2-one
4-{1-[4-(5-propylpyrimidin-2-yl)phenyl]ethyl}morpholine
ethyl 1-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-3-(3-phenylpropyl)piperidine-3-carboxylate
4-chloro-1-methyl-3-{[4-(pyrimidin-4-yl)piperidin-1-yl]methyl}-1H-indazole
(4aR,7aS)-1-propyl-4-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4R)-1-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]-4-phenylpyrrolidine-3-carboxylic acid
N-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-3-(4-methylpiperazine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
8-fluoro-3-[4-(4-methoxybutyl)piperazine-1-carbonyl]-1,4-dihydroquinolin-4-one
1-ethyl-5-({[5-(methylcarbamoyl)furan-2-yl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-[2-methoxy-4-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
1-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
3-[({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)carbamoyl]pyridin-1-ium-1-olate
(1R,5R)-6-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
3-{2-oxo-2-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethyl}imidazolidine-2,4-dione
ethyl 1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidine-4-carboxylate
2-[4-(2,6-dimethoxypyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
(3S,9aR)-8-(3,5-dichlorobenzoyl)-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{4-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
4-[(2,3-dimethoxyphenyl)methyl]-2-[(3-fluorophenyl)methyl]morpholine
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(2-methylphenoxy)azetidin-1-yl]propan-1-one
2-[(2S,3R)-2-amino-3-hydroxybutanoyl]-N-(thiophen-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
(1R,5S)-3-(2-methyl-5-propylpyrimidin-4-yl)-3,8-diazabicyclo[3.2.1]octane
2-(2H-1,3-benzodioxol-5-ylmethyl)-4-[4-(2,2-diphenylethyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-butyl-N-methyl-3-[(2-methyl-5-oxo-1,4-diazepan-1-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-(2,5-dimethoxyphenyl)acetamide
N-[(6-chloropyridin-3-yl)methyl]-2-(methylamino)pyridine-4-carboxamide
(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)(pyridin-2-yl)methanol
2-(2-{[2-(pyridin-4-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one