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N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-(1,1-dioxo-1λ6-thiolan-3-yl)acetamide
N-(2,3-dihydroxypropyl)-2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
1-cyclohexyl-4-(3-methoxypyridine-2-carbonyl)piperazin-2-one
(1R,3R,5S)-3-(4-methoxyphenyl)-8-(5-methylpyrazine-2-carbonyl)-8-azabicyclo[3.2.1]octane
(2R,3R)-3-{4-[(benzylamino)methyl]-1H-1,2,3-triazol-1-yl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(1,1-dioxo-1λ6-thiolan-3-yl)-1H-1,2,4-triazol-3-yl]acetamide
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5,6-dimethyl-2-(trifluoromethyl)pyrimidine
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidine
1-(cyclopropylmethyl)-3-({[(4-fluorophenyl)methyl](methyl)amino}methyl)-3-hydroxypiperidin-2-one
1-{2-[methyl(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amino]ethyl}piperidin-2-one
N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
N-[2-fluoro-5-(4H-1,2,4-triazol-4-yl)phenyl]-4-{[(propan-2-yl)carbamoyl]methyl}piperazine-1-carboxamide
2,6-difluoro-4-methoxy-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
5-{[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}pyridin-2-amine
(3S,7S,8aS)-7-{[(2,5-dimethylphenyl)methyl]amino}-3-[(4-hydroxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
ethyl 5-ethyl-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)sulfamoyl)-N,N-dimethylbenzamide
3-(3-hydroxyquinoxalin-2-yl)-N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)propanamide
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-2-methylphenyl)urea
(9aR)-2-methyl-8-(naphthalene-1-sulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-ethyl-3-(1-methyl-1H-pyrazol-5-yl)-N-(pyridin-4-ylmethyl)propanamide
2-{1-[(1-{5-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-2-amine
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-4-(piperidin-3-yl)benzamide
3-methyl-6-[4-(piperidine-1-carbonyl)piperidin-1-yl]pyridazine
2-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]acetic acid
3-ethyl-8-[2-(morpholin-4-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1-ethyl-5-oxopyrrolidin-3-yl)-2-(4-fluoro-2-methylbenzenesulfonamido)acetamide
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]({[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl})amine
4-[3-(methanesulfonylmethyl)piperidin-1-yl]-5-methylpyrimidin-2-amine
methyl 4-[(E)-2-phenylethenyl]-1H-pyrrole-2-carboxylate
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-5-methyl-N-[2-methyl-2-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
2-amino-7-[4-(thiophen-2-yl)butanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(4-{[(dimethylsulfamoyl)amino]methyl}-4-hydroxyazepan-1-yl)-2-(thiophen-2-yl)ethan-1-one
1-(2H-1,3-benzodioxole-5-carbonyl)-3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine
3-(dimethyl-1,2-oxazol-4-yl)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)propanamide
N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]-2-(pyridin-3-ylmethyl)pyrrolidine-1-carboxamide
5-fluoro-3-methyl-2-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}-1H-indole
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}thiophene-2-carboxamide
2-(2-aminoethyl)-N-[(4-methoxyphenyl)methyl]-N-methylquinazolin-4-amine
2-(3-chloro-4-hydroxyphenyl)-N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)acetamide
5-{1-[(4-butoxyphenyl)methyl]pyrrolidin-2-yl}-3-methyl-1H-1,2,4-triazole
1-(5-chloro-2-methylphenyl)-4-({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine
1-{3-[4-(4-methoxyphenoxy)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-3-(morpholin-4-yl)butan-1-one
4-[2-(4-propanoylphenoxy)acetyl]-1λ6-thiomorpholine-1,1-dione
6-(4-fluorophenyl)-7-methyl-2-(1,4-oxazepane-4-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
(3aR,5R,6S,7aS)-2-(2-methyl-4-phenylpyridine-3-carbonyl)-octahydro-1H-isoindole-5,6-diol
9-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-(1-hydroxyhexan-2-yl)-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-{1-[(6-ethoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]pyrrolidin-3-yl}-N-methylacetamide