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3-acetamido-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
N'-cyclopentyl-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)butanediamide
3-(2,5-dioxoimidazolidin-4-yl)-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}propanamide
4-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-3-yl}benzoic acid
1-(diethylamino)-3-(4-{[(1-hydroxy-2-methylpropan-2-yl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
2-methyl-7-{2-oxa-7-azaspiro[4.5]decan-7-ylmethyl}-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazine
(3ar,6ar)-N-[3-(3-oxopiperazin-1-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(3aR,6aR)-2-acetyl-5-{[5-(3-chlorophenyl)furan-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-methyl-4-(4-{[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]methyl}phenyl)but-3-yn-2-ol
2-(4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}morpholin-3-yl)acetic acid
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
(1R,3S)-3-[ethyl({2-[(4-methylphenyl)sulfanyl]ethyl})carbamoyl]cyclopentane-1-carboxylic acid
(3aS,7aR)-2-[4-(ethylamino)pyrimidin-2-yl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
(3S,4S)-1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
[2-(1-methyl-1H-pyrazol-4-yl)ethyl]({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylpropyl)acetamide
methyl(oxan-4-ylmethyl){[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}amine
2-[3-(piperidine-1-carbonyl)pyrazine-2-carbonyl]-1,2,3,4-tetrahydroisoquinoline
4-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenol
methyl (2S,4R)-4-(2-cyclopropylquinoline-4-amido)-1-[(2,6-difluorophenyl)methyl]pyrrolidine-2-carboxylate
8-[2-(benzyloxy)benzoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-ethyl-N-(2-methylprop-2-en-1-yl)-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-(4-methoxybenzoyl)piperidine-4-carboxamide
2-(2-chlorophenyl)-2-hydroxy-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
7-[2-hydroxy-3,5-bis(propan-2-yl)benzoyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(2,4-dihydroxyphenyl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
(1R,5R)-3-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
4-ethyl-3-[1-(1-propyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[4-(propan-2-yloxy)phenyl]-3-(pyrrolidine-1-carbonyl)pyridine
1-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
2-[methyl({4-methyl-5-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
3-chloro-N-[(1-ethyl-1H-imidazol-5-yl)methyl]-4-fluoro-1-benzothiophene-2-carboxamide
1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-(2H-indazol-2-yl)ethan-1-one
[1-({1-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
1-(1-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,6-tetrahydropyridin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-[3-(3-methylphenoxymethyl)piperidin-1-yl]ethan-1-amine
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)(1,3-thiazol-2-ylmethyl)amine
4-(ethoxymethyl)-N-[3-(3-fluorophenyl)phenyl]piperidine-1-carboxamide
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
5-({[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}methyl)-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]-2-(1H-1,2,3-triazol-1-yl)acetamide
N,2-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}thieno[2,3-d]pyrimidin-4-amine
(4aR,8aS)-1-[(3-fluorophenyl)methyl]-6-(furan-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-(2-methoxybutanoyl)-N-[(5-methylfuran-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-{4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperazin-1-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]-N-[2-(1H-pyrazol-4-yl)ethyl]pyridin-2-amine
4-[(2-{1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)methyl]pyridine
[1-(3-methoxybenzenesulfonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol