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9-(4-methyl-1,3-thiazole-5-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(3S)-3-hydroxypyrrolidin-1-yl]-N-(2-methanesulfonylethyl)-1-methyl-1H-1,3-benzodiazole-5-carboxamide
4-[9-(1,2,3,6-tetrahydropyridin-1-yl)-3-azaspiro[5.5]undecane-3-carbonyl]benzonitrile
ethyl 2-{[2-(dimethylamino)ethyl]carbamoyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxylate
2-methoxy-1-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)ethan-1-one
2-[1-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]pyridine
methyl (2R,4S)-4-hydroxy-1-(2-methoxyacetyl)piperidine-2-carboxylate
(2S,3R)-2-[(3-{[(4-fluorophenyl)methyl]amino}phenyl)formamido]-3-hydroxybutanamide
1-methyl-4-[(5-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazol-3-yl)methyl]piperazine
2-[6-(dimethylamino)pyridine-3-carbonyl]-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one
2-methyl-6-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
1-(1-methyl-1H-pyrazole-5-carbonyl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
3-{[3-(methylcarbamoyl)propyl]sulfamoyl}-N-(oxolan-3-yl)benzamide
1-[(4-fluorophenyl)methyl]-4-{[2-(methylsulfanyl)phenyl]methyl}-1,4-diazepane
N-[3-(furan-2-yl)phenyl]-1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]piperidine-4-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[3-(pyridin-4-yl)azetidin-1-yl]ethan-1-one
6-{[2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-cyclopentyl-5-[(3-methylthiophen-2-yl)sulfonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-methyl-9-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
(1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methanol
N-{4-[({[4-(hydroxymethyl)oxan-4-yl]methyl}(methyl)amino)methyl]phenyl}acetamide
3-[(1-methanesulfonylpiperidin-3-yl)methyl]-1-{3-[(2-methylprop-2-en-1-yl)oxy]phenyl}urea
N-({5-[(4-methyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
(1S,6R)-9-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propanoyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
(3S,4S)-1-[2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
7-{2-[2-(2-methylpropyl)-1H-1,3-benzodiazol-1-yl]propanoyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(2S,4S)-4-(2,3-dihydro-1-benzofuran-5-amido)-N-ethyl-1-(3-methylbut-2-en-1-yl)pyrrolidine-2-carboxamide
N-[2-(furan-2-yl)ethyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
N-(3,5-dimethoxyphenyl)-4-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}benzamide
2,6-dimethoxy-3-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
1-methyl-3-(3-phenyl-1,2,4-thiadiazol-5-yl)-1-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}urea
4-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidine
1-[4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperidin-4-ol
3-propoxy-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidine
3-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]piperidine-1-carboxamide
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-(3-chlorophenyl)-2-hydroxy-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}acetamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-methyl-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
N-methyl-4-(2-methyl-1H-imidazol-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)butanamide
1-[(2-methylphenyl)methyl]-5-{spiro[2.3]hexan-1-yl}-1H-1,2,4-triazole
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5-(oxolan-2-yl)thiophene-2-carboxamide
2-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
1-methyl-6-{[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-4-one
N-(1,4-dioxan-2-ylmethyl)-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyridine-3-carboxamide
methylbis(quinolin-2-ylmethyl)amine
8-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-chloro-3-fluoro-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyridin-2-amine