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1-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]-2-(5-chloro-6-methyl-1-benzofuran-3-yl)ethan-1-one
N-ethyl-2-[4-(2-methyl-3-phenylcycloprop-2-ene-1-carbonyl)piperazin-1-yl]acetamide
N,3-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]furan-2-carboxamide
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
5-(2-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-2-oxoethyl)-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(5-acetylthiophene-3-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
6-cyclopentyl-2-(4-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
3-methyl-N-{1-[1-(3-phenoxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
N-(1-{5-[(cyclohexylmethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)furan-3-carboxamide
2-(pyridin-3-ylmethyl)-8-(quinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
6-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoline
(4aS,8aR)-6-[2-(methylamino)-1,3-thiazole-4-carbonyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-methyl-2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-[(2S)-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethan-1-one
2-[(methylcarbamoyl)methyl]-N-[3-(methylsulfanyl)phenyl]-3-oxopiperazine-1-carboxamide
(4aS,7aR)-1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4aS,7aR)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(3-methylbutyl)piperazin-2-one
1-{[2-(3-chlorophenyl)-7-fluoroquinolin-3-yl]methyl}piperidin-4-ol
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-N-(propan-2-yl)-2,3,4,9-tetrahydro-1H-carbazole-7-carboxamide
4-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}thiomorpholine
phenyl (3S,9R)-2,8-dioxo-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-11-carboxylate
1-(2H-1,3-benzodioxol-5-ylmethyl)-5-[(4-methanesulfonylphenyl)methyl]-1H-1,2,4-triazole
3-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-6-methylpyridazine
methyl (1S,3S,3aR,6aS)-3-(1,3-dimethyl-1H-pyrazol-4-yl)-1-(hydroxymethyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
(3S,4S)-N,4-bis(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidine-1-carboxamide
(benzylsulfamoyl)[2-(dimethyl-1,3-thiazol-2-yl)ethyl]amine
N-[2-(4-methoxyphenyl)phenyl]-1-(3-methylbut-2-en-1-yl)piperidine-3-carboxamide
N-[(5-chloro-2-propoxyphenyl)methyl]-2-(2-oxopiperidin-1-yl)acetamide
1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-3-[3-(propan-2-yloxy)benzoyl]piperidine
(2R,3R,6R)-5-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-(5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1H-pyrazol-3-yl)pyridine
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-(pyridin-2-yl)propanamide
5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
3-methyl-1-(2-methylpropyl)-4-[3-(morpholin-4-yl)benzoyl]piperazin-2-one
N-{5-chloro-2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carbonyl]phenyl}propanamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]benzamide
2-{4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
6-{[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}pyridine-2-carboxylic acid
N-methyl-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
N-cyclopropyl-5-(1H-indole-2-carbonyl)-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{4-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidine-1-carbonyl]piperidin-1-yl}ethan-1-one
2-(4-fluorophenyl)-1-(furan-3-carbonyl)piperidine
N-(1,3-dihydroxypropan-2-yl)-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[2-(isoquinolin-5-yl)pyridin-4-yl]methanol
3-(2-fluorophenyl)-3-{[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]formamido}propanoic acid
[(2-fluorophenyl)methyl][(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl](2-methoxyethyl)amine