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1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
N-[(4-fluorophenyl)methyl]-1-methyl-5-{[(3-methyl-1,2-oxazol-5-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-({2-[5-(piperidine-1-carbonyl)pyridin-2-yl]phenyl}methyl)morpholine
methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})(thiophen-2-ylmethyl)amine
(3R,4S)-4-[({2-[(2-chloro-6-fluorophenyl)methoxy]phenyl}methyl)(methyl)amino]oxolan-3-ol
1,3-dimethyl-2,6-dioxo-N-[2-(thiophen-2-yl)ethyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(2S)-2-({1-[(diethylcarbamoyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)-3-methylbutanamide
N-(1-methyl-1H-pyrazol-5-yl)-2-{3-[4-(morpholin-4-ylmethyl)thiophen-2-yl]-1H-pyrazol-1-yl}acetamide
4-[3-(propan-2-yl)-1H-pyrazol-5-yl]-1-(1H-pyrrole-2-carbonyl)piperidine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(1-hydroxycyclopentyl)ethyl]benzamide
N-(4-chloro-3-methylphenyl)-2-({[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)acetamide
3-[1-(2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)piperidin-3-yl]benzoic acid
3-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole
2-(azepan-1-yl)-N-[(2-phenoxypyridin-3-yl)methyl]acetamide
3-{[5-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2-oxazole
N-ethyl-2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl){[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
3-{[(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}-4H-chromen-4-one
6-cyclopentyl-3-(oxolan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
4-(4-fluorophenyl)-N-(oxan-2-ylmethyl)-4-oxobutanamide
6-(2-hydroxy-5-methoxyphenyl)-2-[3-(pyrrolidin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
(3R,5S)-5-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine-1-carbonyl]pyrrolidin-3-amine
3-{2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}-3,4-dihydroquinazolin-4-one
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N,2,6-trimethyl-N-[3-(oxolan-2-yl)propyl]quinoline-3-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-{[(3-hydroxy-4-methoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
1-[4-(2-chlorophenoxy)piperidin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
1-benzyl-4-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]piperazine
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-2-[3-methyl-1-(3-methylphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-methyl-4-(piperidin-1-ylmethyl)-N-[2-(pyridin-2-yl)ethyl]benzamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidin-3-yl]furan-3-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(5-butylthiophen-2-yl)methyl]-N-ethylpyrrolidine-3-carboxamide
5-chloro-4,6-dimethyl-2-oxo-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-1,2-dihydropyridine-3-carboxamide
1-[1-(3,5-dimethylbenzoyl)piperidin-3-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
3-(3,5,5-trimethylcyclohex-2-en-1-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(2-ethylphenoxy)ethyl]-N-methyl-1,1-dioxo-1λ6-thiane-4-carboxamide
5-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
(3aR,6aR)-2-benzoyl-5-cyclobutanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
{1-[2-({7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)ethyl]piperidin-2-yl}methanol
{5-[(2-aminopyridin-3-yl)methyl]-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
benzyl({[3-(cyclohexyloxy)-2-hydroxypropyl]sulfamoyl})amine
dimethyl(3-{2-[1-(1-phenylcyclopropanecarbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
3-(1,5-dimethyl-1H-pyrazol-4-yl)-1-[(2-methylphenyl)methyl]-1-(oxolan-2-ylmethyl)urea
5-(2-methylpropyl)-1'-[(1-propyl-1H-imidazol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-{2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}propanamide