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7-(2,2-dimethylpropyl)-2-[(2-phenyl-1,3-oxazol-4-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-(2,6-dimethylphenoxy)-1-(4-fluoro-2-methylbenzoyl)azetidine
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-[2-(furan-2-yl)ethyl]-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
5-(2-methoxy-4-methylbenzoyl)-3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine
1-(naphthalen-2-yl)-4-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperazine
(3aS,6aS)-2-(oxan-4-yl)-5-(pyrimidin-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(oxolan-2-ylmethyl)-N-[4-(1H-1,2,4-triazol-1-yl)phenyl]piperazine-1-carboxamide
2-methoxy-3-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
(1R,5R)-3-(4-ethyl-5-methylthiophene-3-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-{3-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
3-(2-methyl-1H-imidazol-1-yl)-1-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
(4-{[4-(morpholine-4-sulfonyl)phenyl]methyl}-1,4-oxazepan-6-yl)methanol
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5-(cyclooctylamino)azepan-2-one
2-(dimethylamino)-N-[(5-ethylpyridin-2-yl)methyl]-N,4-dimethylpyrimidine-5-carboxamide
(4aR,7aS)-1-ethyl-4-[2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[2-(propan-2-yloxy)-5-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)phenyl]methanol
3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-[1-(4-phenylbutanoyl)piperidin-4-yl]-5-propylimidazolidine-2,4-dione
2-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}-3-(propan-2-yl)urea
(3aR,7aS)-2-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
3-chloro-6-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}pyridine-2-carboxylic acid
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
4-{7-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfamoyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}-4-oxobutanamide
3-[(dimethylamino)methyl]-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4,4-difluoropiperidine
(3aR,6aR)-2-cyclopentyl-5-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{1-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]piperidin-4-yl}-1,3-oxazolidin-2-one
N-benzyl-4-(quinolin-6-yloxy)piperidine-4-carboxamide
1-[(4-fluorophenyl)methyl]-5-(2-methoxy-5-methylbenzoyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
2-(3-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
1-[(3-fluorophenyl)methyl]-4-(5-phenyl-1,2,4-oxadiazol-3-yl)piperazine
N-[4-(3-chloropyridin-2-yl)phenyl]methanesulfonamide
4-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
[(5-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}thiophen-3-yl)methyl]dimethylamine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-(4-methylphenoxy)piperidine-4-carboxamide
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1H-1,2,3-triazole-5-carboxamide
N,N-dimethyl-6-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}pyridine-3-carboxamide
7-[3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
5-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidine-1-carbonyl}-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
3-(3-fluorophenyl)-4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperazin-2-one
5-{5-[1-ethyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
(4aS,8aR)-1-(3-aminopropyl)-6-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-decahydro-1,6-naphthyridin-2-one
3-[4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperazin-1-yl]phenol
2-{8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-6-methylpyridine-3-carbonitrile
(3S,4R)-N,N-dimethyl-4-(propan-2-yl)-1-(1H-pyrrole-2-carbonyl)pyrrolidin-3-amine