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2-ethyl-8-(2-methyl-5-propylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
3-[(dimethylamino)methyl]-1-(2-phenylquinoline-4-carbonyl)pyrrolidin-3-ol
2-cyclopropyl-3-oxo-N-[2-(propan-2-yl)phenyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-(2-ethylphenyl)-3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carboxamide
ethyl 4-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}piperazine-1-carboxylate
4-ethyl-5-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-1,3-thiazol-2-amine
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-3-(1,2-oxazinan-2-yl)propanamide
5-(1,3-benzothiazol-2-ylmethyl)-1-(cyclopropylmethyl)-N-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[1-(1-methylpiperidin-4-yl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-N-[(1R)-1-phenylethyl]pyrimidin-2-amine
ethyl 1-[2-chloro-5-(trifluoromethyl)benzoyl]-4-(cyclopropylmethyl)piperidine-4-carboxylate
5-{[2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]sulfonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-{3-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1H-pyrazol-1-yl}acetamide
2-(4-fluorophenyl)-N-[2-(7-{[5-(methoxymethyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]acetamide
1-[2-(1H-imidazol-4-yl)ethyl]-2-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-1H-imidazole
2-(1,2-benzoxazol-3-yl)-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-N-methylacetamide
(3S,4S)-3-hydroxy-4-[(1H-imidazol-2-ylmethyl)(methyl)amino]-1λ6-thiolane-1,1-dione
3-cyclopropyl-1-(2-phenylethyl)-5-[1-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazole
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decane
1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-[2-(2-methylpropanesulfonyl)ethyl]urea
2-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}phenoxy)ethan-1-ol
5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-(1,2-oxazol-3-ylmethyl)pyridin-2-amine
(2S,4R)-N-methyl-1-(oxan-4-yl)-4-{4H-thieno[3,2-b]pyrrole-5-amido}pyrrolidine-2-carboxamide
3-(4-chlorophenyl)-4-[(3-propyl-1H-pyrazol-5-yl)formamido]butanoic acid
2-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
1-{4-[hydroxy(pyridin-2-yl)methyl]piperidin-1-yl}-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
N-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1-(pyridin-3-ylmethyl)piperidin-4-amine
1-[1-(6-methylpyridazin-3-yl)piperidin-4-yl]piperidin-3-ol
methyl[3-(methylsulfanyl)butyl]{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
3-(3-methylphenyl)-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidine
3-(2-phenylethyl)-5-{1-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazole
8-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
3-ethyl-5-({2-[2-(methylsulfanyl)phenyl]-1H-imidazol-1-yl}methyl)-1,2-oxazole
4-(1-butyl-1H-imidazol-2-yl)-1-(5-fluoro-2-methylbenzoyl)piperidine
2-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]pyridine-4-carboxylic acid
1-(3,5-difluorophenyl)-N-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-methyl-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-1H-1,3-benzodiazole-5-carboxamide
[(3-{[1-(2,1,3-benzothiadiazole-4-sulfonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(thiophen-2-ylmethyl)amine
N-[1-(3,4-dimethoxyphenyl)ethyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(3S)-1-[3-(3-fluorophenyl)benzoyl]pyrrolidin-3-yl]acetamide
1-[(1S,5R)-6-(2,5-dimethylbenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
7-methyl-2-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-2,7-diazaspiro[4.5]decan-6-one
4-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}phenol
4-[4-(3-methoxypiperidin-1-yl)piperidin-1-yl]-6-methyl-2-(pyrrolidin-1-yl)pyrimidine
5-[ethyl(2-methylprop-2-en-1-yl)amino]-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-({3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]phenyl}amino)acetic acid
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,1,3-trimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-N-{[4-(methylsulfanyl)phenyl]methyl}cyclopropanamine