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4-hydroxy-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
5-(3-fluorophenoxymethyl)-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]-1H-pyrazole-3-carboxamide
N-(4-{[cyclopentyl(prop-2-en-1-yl)carbamoyl]methyl}phenyl)butanamide
2-chloro-4-{[ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}-6-methoxyphenol
3-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]-1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
3-{[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl](methyl)amino}-N-methylpropanamide
5-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
({4-ethyl-5-[1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-(3-{1-[(3-cyanophenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}-1-methyl-1H-pyrazol-5-yl)acetamide
N-{[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]methyl}-4-phenylbenzamide
2-{[(1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidin-3-yl)oxy]methyl}pyridine
2-cyclopropyl-8-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one
N-(2,3-dihydro-1H-inden-1-yl)-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
2-(7-methyl-1H-indol-3-yl)pyridine-4-carboxamide
4-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-1,4-oxazepan-6-ol
2-[3-(2-fluorophenyl)-1H-pyrazol-1-yl]-N-(1-propyl-1H-indazol-3-yl)acetamide
3-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-3-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
2-[4-(1H-pyrazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
7-[2-(methylamino)pyridine-3-carbonyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{[3-(4-carboxyphenyl)piperidin-1-yl]sulfonyl}piperidine-4-carboxylic acid
3-[1-(3-cyclopentylpropyl)piperidin-4-yl]-N-cyclopropylpropanamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(4-methyl-1H-imidazole-2-carbonyl)pyrrolidin-3-yl]methanol
(1R,3S)-3-(2-aminoethoxy)-7-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)-7-azaspiro[3.5]nonan-1-ol
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
3-methyl-5-{1-[(4-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-2-yl}-1H-1,2,4-triazole
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-(thiophen-2-ylmethyl)benzamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(3-methylphenyl)methyl]pyrrolidin-3-yl]methanol
2-{[(2-methoxybutyl)amino]methyl}-6-methylquinolin-4-ol
(3-{2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-ylmethyl]phenoxy}propyl)dimethylamine
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-ethyl-N-[(3-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)pyrimidine-5-carboxamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
N,2,6-trimethyl-N-[1-(1,3-thiazol-2-yl)ethyl]pyrimidine-4-carboxamide
2-{2-[(4-fluorophenyl)methyl]morpholin-4-yl}ethan-1-ol
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-(naphthalen-2-ylmethyl)-1,4-diazepan-5-one
N-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methoxy]phenyl}propanamide
2-(4-{pyrazolo[1,5-a]pyridine-3-carbonyl}morpholin-3-yl)acetic acid
(3aS,6aS)-2-[(2-phenoxyphenyl)carbamoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[4-(oxan-2-ylmethoxy)phenyl]-3-[2-(pyridin-3-yl)ethyl]urea
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(2-oxopropanoyl)piperidine-4-carboxamide
1-[4-(6-amino-4-methylpyridin-3-yl)phenyl]-3,3-dimethylurea
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
(1S,9aR)-1-{[4-(1,3-benzothiazol-2-yl)-1,4-diazepan-1-yl]methyl}-octahydro-1H-quinolizine
2-[4-(3,5-dichlorobenzamido)-3,5-dimethyl-1H-pyrazol-1-yl]acetic acid
(2-{2-[1-(3-ethoxybenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]oxolane-3-carboxamide
N-methyl-5-oxo-1-(pyridin-2-ylmethyl)-N-(thian-4-yl)pyrrolidine-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,4-dimethylpyrimidin-2-amine
5-(3-benzyl-1H-1,2,4-triazol-5-yl)-1H-1,3-benzodiazole
N-cyclopropyl-3-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]propanamide