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4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-2-(propan-2-yl)pyrimidine
1-(3-benzoylpiperidin-1-yl)-2-(thiophen-2-yl)ethan-1-one
2-(dimethylamino)-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-2-(3-methylphenyl)acetamide
N,N-dimethyl-2-{methyl[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amino}acetamide
2-(dimethylamino)-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)acetamide
3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3-ethyl-1-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]urea
3-methyl-4-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-1-(2-methylpropyl)piperazin-2-one
N-({1-[(6-methoxy-2H-chromen-3-yl)methyl]piperidin-4-yl}methyl)propanamide
3-tert-butyl-N-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-methyl-1H-pyrazole-5-carboxamide
2-(1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-amine
3-(1H-1,3-benzodiazol-1-yl)-1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
2-amino-8-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
(2S,4R)-4-[(1-benzylpiperidin-4-yl)amino]-1-[(3-chlorophenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)piperidin-4-ol
4-{[5-(2-fluoro-4,5-dimethoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]methyl}pyridine
4-(4-chloro-2-methoxy-5-methylphenyl)-4H-1,2,4-triazole
4-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}thiomorpholine
N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-1-phenylpiperazine-2-carboxamide
2-(4,5-dimethyl-1H-imidazol-1-yl)-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)acetamide
1-({5-[(4-methoxy-2-methylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
3-({1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1H-pyrazole
3-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-1-(2,3,4-trifluorophenyl)urea
3-(2-methyl-2-phenylpropanoyl)-3,9-diazaspiro[5.6]dodecan-10-one
methyl 2-{1-[1-(2-fluorophenyl)cyclopropanecarbonyl]-3-oxopiperazin-2-yl}acetate
N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-4-(trifluoromethyl)pyrimidin-2-amine
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
2-amino-3-ethyl-N-[2-(pyridin-2-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-methyl-5-{4-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(3-methoxybenzoyl)piperidine
N-butyl-2-(1-methyl-1H-pyrrol-2-yl)-2-oxo-N-(thiophen-3-ylmethyl)acetamide
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-3-(1-methylpiperidin-2-yl)propanamide
5-benzyl-4-(furan-3-ylmethyl)-1-(3-methoxyphenyl)piperazin-2-one
methyl 3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-3-yl]propanoate
2-({5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazol-3-yl}formamido)-N-(propan-2-yl)acetamide
N-[4-(2,2-dimethylpropanamido)-3-methoxyphenyl]-N'-(2-ethylphenyl)ethanediamide
2-amino-8-{3-[(diethylamino)methyl]-4-methoxyphenyl}-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
3-methyl-7-(2,3,4,9-tetrahydro-1H-carbazole-6-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-[(4-{5-[(cyclohexylmethyl)sulfanyl]-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]phenol
N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
2-[4-(2-methylpyrimidin-4-yl)piperidine-1-carbonyl]pyridin-3-ol
N-[(1-methylpyrrolidin-3-yl)methyl]-2,2-diphenylacetamide
[(3aS,6aS)-2-(8-fluoroquinoline-2-carbonyl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]acetamide
1-ethyl-N-[(6-methylpyridin-2-yl)methyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-yl]-2-ethoxyethan-1-one
N-(5-methyl-1,2-oxazol-3-yl)-N'-[(2E)-3-phenylprop-2-en-1-yl]-N'-propylethanediamide
5-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
1-{2-oxo-2-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}imidazolidine-2,4-dione
2-[1-cyclohexyl-5-(2-methoxypyridin-3-yl)-1H-1,2,4-triazol-3-yl]acetamide