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1-cyclohexyl-4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-2-one
N-[3-(furan-2-yl)propyl]-2-methyloxane-2-carboxamide
3-[N-(propan-2-yl)-1-(2,2,3,3-tetramethylcyclopropyl)formamido]propanamide
1-{[3-fluoro-2-(trifluoromethyl)phenyl]methyl}azepan-2-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carboxamide
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
5-ethyl-4-(pyrrolidin-1-ylmethyl)-N-[2-(1H-1,2,4-triazol-1-yl)propyl]furan-2-carboxamide
[3-(2-methoxyethyl)-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-3-yl]methanol
methyl (2S,4R)-1-methyl-4-[3-(1,2-oxazolidin-2-yl)propanamido]pyrrolidine-2-carboxylate
N-cyclohexyl-4-[6-(1-hydroxyethyl)pyridin-2-yl]benzene-1-sulfonamide
2-{[(4-methyl-1H-imidazol-5-yl)methyl][(2-methylphenyl)methyl]amino}butan-1-ol
N4-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-6-(propan-2-yl)pyrimidine-2,4-diamine
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-4-oxo-1,4-dihydroquinoline-2-carboxamide
4-[4-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](methyl)amino}methyl)phenyl]-2-methylbutan-2-ol
5-(propan-2-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1,2-oxazole-3-carboxamide
methyl[(3-methyl-1,2-oxazol-5-yl)methyl]{[3-(1H-1,2,4-triazol-5-yl)phenyl]methyl}amine
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-3-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(furan-3-carbonyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
4-phenyl-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}azepane
4-(5-chloro-2-methylphenyl)-3-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one
9-(5-hydroxypyrazine-2-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,7S,8aS)-3-(2-methylpropyl)-7-[(thiophen-3-ylmethyl)amino]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-(9H-purin-6-yl)piperidin-3-ol
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
1-[4-(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,2,3,6-tetrahydropyridin-4-yl)-1H-pyrazol-1-yl]butan-2-ol
N-[(1R,2R)-2-acetamido-2,3-dihydro-1H-inden-1-yl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
2-methyl-4-{4-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]phenyl}butan-2-ol
6-fluoro-4-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
[(2-chloro-6-fluorophenyl)methyl](ethyl){[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
(furan-2-ylmethyl)({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})[2-(morpholin-4-yl)ethyl]amine
(1S,6R)-3-methyl-9-(thiophene-2-sulfonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
methyl 2-[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidine-1-carbonyl]benzoate
N-(1,4-dioxan-2-ylmethyl)-5-(1H-indol-1-ylmethyl)-N-methyl-1H-pyrazole-3-carboxamide
4-(piperidin-1-yl)-1-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-yl)butan-1-one
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-5-(methoxymethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
methyl 3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[(3-methylphenyl)methyl]piperidin-3-yl]propanoate
N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-3-(pyrrolidin-1-yl)propan-1-one
4-(2-chloro-4-methoxyphenoxy)-1-(dimethylcarbamoyl)piperidine-4-carboxylic acid
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[3-(methylsulfanyl)propyl]piperidine
1-cyclohexyl-N-(2-hydroxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-[(5-methylfuran-2-yl)methyl]piperazin-2-one
1-[1-(2-aminopyridine-4-carbonyl)piperidin-4-yl]-N-cyclopropyl-1H-1,2,3-triazole-4-carboxamide
3-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydroquinoxalin-2-one
methyl({2-methylimidazo[1,2-a]pyridin-3-yl}methyl){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-N-(2-methylpropyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
(4S)-4-phenyl-3-(pyrimidin-2-ylmethyl)-1,3-oxazolidin-2-one
1-[4-(furan-2-ylmethoxy)phenyl]-3-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
N-(adamantan-1-yl)-4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-{2-chloro-4-[2-(pyridin-2-yl)-1H-imidazol-1-yl]phenoxy}acetic acid