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1-[2-(4-fluorophenyl)piperidin-1-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-phenylethyl)acetamide
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}acetamide
(4aR,8aR)-4-[(5-ethylfuran-2-yl)methyl]-octahydro-2H-1,4-benzoxazine
4-[5-({4-[(1S,2S)-2-hydroxycyclohexyl]piperazin-1-yl}methyl)-1,2,4-oxadiazol-3-yl]benzoic acid
N-[1-(pyridin-4-yl)propan-2-yl]-4-sulfamoylbenzamide
N-methyl-2-(1-methylcyclopropanecarbonyl)-N-(propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-methyl-5-propylpyrimidine
2-(dimethyl-1,3-thiazol-5-yl)-N-{[8-(propan-2-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
3-{2-[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
5-amino-4-chloro-N-[3-(1H-indazol-1-yl)propyl]-1H-pyrazole-3-carboxamide
ethyl 2-[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]-1,3-oxazole-4-carboxylate
1-(oxane-2-carbonyl)-2,2-bis(prop-2-en-1-yl)pyrrolidine
(2R,3R)-1'-(1-benzofuran-5-ylmethyl)-3-(dimethylamino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-[5-({1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}methyl)thiophen-2-yl]-2-methylbut-3-yn-2-ol
(3R,4R)-1-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]-3,4-dimethylpyrrolidin-3-ol
{1-[({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}(methyl)amino)methyl]cyclobutyl}methanol
(4aR,7aS)-1-(cyclopropylmethyl)-4-[2-(phenylsulfanyl)ethyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(5-{[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
2-cyclopropyl-1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)ethan-1-one
N-[(1S,2R)-2-aminocyclobutyl]-3-[(4-fluorophenyl)formamido]propanamide
(1R,7S)-6-(4-methyl-1,4-diazepane-1-carbonyl)-3-(pentan-3-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[3-(pyridin-4-yl)propyl]benzamide
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
11-[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
N-(6-chloropyridin-3-yl)-4-[(dimethylamino)methyl]-4-hydroxyazepane-1-carboxamide
1-(furan-2-ylmethyl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
2-(3-methoxyphenyl)-N-methyl-N-[2-(4-methylpiperidin-1-yl)ethyl]acetamide
5-cyclopropyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-ethyl-3-(oxan-4-ylmethyl)-1-{4-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}urea
7-(1-benzothiophen-3-yl)-4-(2,4-dimethoxybenzoyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-(piperidin-1-yl)piperidine-4-carboxamide
5-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
4-({[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}amino)-N-ethylpiperidine-1-carboxamide
5-[(4-methyl-3-phenylpiperazin-1-yl)methyl]-2-(propan-2-yl)pyrimidine
7-(2-oxoimidazolidin-1-yl)-4-(6-phenoxypyridin-3-yl)-1,2,3,4-tetrahydroquinolin-2-one
3-(1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-1-(pyrrolidin-1-yl)propan-1-one
2-(hydroxymethyl)-N-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-1H-1,3-benzodiazole-5-carboxamide
(1R,9S)-5-amino-3-[4-(1H-imidazol-1-yl)phenyl]-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
9-[2-(pyridin-4-yl)ethanesulfonyl]-3,9-diazaspiro[5.6]dodecane
(2R,4S)-1-(3-chloro-4-hydroxybenzoyl)-4-hydroxypiperidine-2-carboxylic acid
1-{2-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]pyrimidin-4-yl}piperidin-4-ol
1-[7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]piperidin-4-amine
2-methyl-2-[4-(4-methylphthalazin-1-yl)phenyl]propanenitrile
4-benzyl-3-ethyl-1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-1,4-diazepan-5-one
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-ethyl-2-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1,3-thiazole-5-carboxamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide