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(5S)-5-[({[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]pyrrolidin-2-one
2-{[(4-fluorophenyl)methyl](methyl)amino}-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]ethan-1-one
N-[4-(3-methylphenyl)phenyl]-1-[(2S)-oxolane-2-carbonyl]piperidine-4-carboxamide
N-benzyl-3-{[1-(pyrimidin-2-yl)piperidin-4-yl]oxy}benzamide
4-{2-[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]ethyl}-4H-1,2,4-triazole
2-(3-chloro-4-methylbenzenesulfonyl)-2,8-diazaspiro[4.5]decane
2-(dimethylamino)-N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}benzamide
3-[(3R,4S)-4-(dimethylamino)-1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-3-yl]propan-1-ol
9-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(2-chlorophenyl)methyl]-3-[1-(1H-indole-5-carbonyl)piperidin-3-yl]propanamide
(5S,9aS,9bS)-5-(1,3-diphenyl-1H-pyrazol-4-yl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{[5-(4-fluorophenyl)furan-2-yl]methyl}-3-(1-methylpiperidin-3-yl)propanamide
[1-(1H-indol-1-yl)propan-2-yl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-methoxyethan-1-one
1-[3-phenyl-3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propyl]-1H-1,2,4-triazole
3-(4-benzylpiperazine-1-carbonyl)-2-(cyclopentylmethyl)-6-methyl-1-(pyridin-3-ylmethyl)-1,4-dihydropyridin-4-one
2-amino-N-[(3R,4S)-4-cyclopropyl-1-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]pyrrolidin-3-yl]acetamide
7-[3-(4-hydroxyphenyl)propanoyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
8-[2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetyl]-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2R,3S,6R)-3-phenyl-5-(1,3-thiazol-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-4-[(2-methyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
N-[3-(4-methoxyphenyl)propyl]-6-(2-methylpyrrolidin-1-yl)pyridine-3-carboxamide
4-(1,3-benzothiazole-6-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
1-(1,2,3,4-tetrahydroisoquinolin-2-yl)-3-[3-({[2-(1,3-thiazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-{1-[1-(5-fluoro-1H-indole-2-carbonyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N,3-dimethylbutanamide
N-(2-oxoazepan-3-yl)-3-(1H-pyrazol-1-yl)benzamide
N-(2-acetamidophenyl)-2-{[(1S)-1-phenylpropyl]amino}acetamide
[(3R,4R)-1-(2-methyl-1,3-thiazole-5-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
4-ethyl-1-methyl-3-({1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-(thiophen-3-ylmethyl)acetamide
4-(piperidin-3-yl)-N-[(4-sulfamoylphenyl)methyl]benzamide
2-(4-{[5-(3-methoxypropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}piperazin-1-yl)pyrazine
(1-methyl-5-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
N-(1-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methylbenzamide
(2S)-N2-[(3-fluoro-4-methoxyphenyl)methyl]pyrrolidine-1,2-dicarboxamide
5-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-1-[(2-methoxyphenyl)methyl]piperidin-2-one
2-amino-8-(quinolin-8-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
2-[4-(1H-imidazol-2-ylmethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl]acetic acid
1-[2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carbonyl]-4-methylpiperidine
{4-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenyl}methanol
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1H-indole-2-carbonyl)piperazin-2-one
1-{[1-(1-cyclobutylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl}azepane
N-(2-methyl-1-benzofuran-7-yl)-4-(4-methyl-1H-pyrazol-3-yl)piperidine-1-carboxamide
N-(2,3-dihydro-1H-inden-1-yl)-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
2-[3-(4-ethoxyphenyl)-4-methoxyphenyl]ethan-1-amine
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
1-(3-hydroxypropyl)-3-(1-methyl-1H-1,2,3-triazol-4-yl)-1-[(2E)-3-phenylprop-2-en-1-yl]urea
(2S,4S)-4-cyclopropaneamido-N-ethyl-1-[2-(propan-2-yl)pyrimidine-5-carbonyl]pyrrolidine-2-carboxamide
2-(cyclohexylmethyl)-4-[(trimethylpyrazin-2-yl)methyl]morpholine