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(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(6-methylpyridazin-3-yl)pyrrolidin-3-amine
N-(4-fluorophenyl)-1-(3-hydroxypropanoyl)piperazine-2-carboxamide
N-(4-{2-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]acetamido}phenyl)-N-methylacetamide
N4-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-N2,6-dimethylpyrimidine-2,4-diamine
2-(4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)ethan-1-ol
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[2-(thiophen-3-yl)acetyl]piperidin-3-yl}propanamide
9-(1-benzofuran-5-carbonyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
8-methoxy-3-[2-(piperazin-1-yl)ethyl]-3,4-dihydroquinazolin-4-one
8-(2-methoxy-4-methylbenzenesulfonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-{2-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidine-1-carbonyl]phenyl}-1λ6-thiomorpholine-1,1-dione
1-{1-[(4-methanesulfonylphenyl)methyl]piperidin-3-yl}pyrrolidin-2-one
2-(adamantan-1-yl)-4-hydroxy-N-[2-(1H-imidazol-1-yl)ethyl]pyrimidine-5-carboxamide
1-[2-(2H-1,3-benzodioxol-5-ylformamido)ethyl]-N-(2-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-(2-oxopyrrolidin-3-yl)benzamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2-methyl-1,8-naphthyridine-3-carboxamide
N-{2-[4-(4-methyl-1,4-diazepane-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}adamantane-1-carboxamide
2-cyclopropyl-N,N-dimethyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecane-9-sulfonamide
6-ethyl-1-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(dimethyl-1,2-oxazol-4-yl)-1-[4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
8-benzyl-3-[2-(dimethylamino)ethyl]-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)acetamide
(4aS,7aR)-1-(azepane-1-sulfonyl)-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(3-fluorophenyl)-N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
N-[(4-fluorophenyl)methyl]-5-[(1-hydroxy-2-methylpropan-2-yl)amino]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(3-methylpyridin-2-yl)methyl]-4-(2-methylpyrrolidine-1-carbonyl)benzene-1-sulfonamide
4-(pyrazine-2-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[methyl(2-phenylethyl)amino]-N-[(3-methylpyridin-4-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-2,3-dimethylbenzene-1-sulfonamide
N-[(4-methoxyphenyl)methyl]-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
4-{5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carbonyl}-1-methylpiperazin-2-one
3-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
3-{1-methyl-4-[3-(1H-pyrazol-1-yl)azetidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
4-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]pyridin-2-amine
{[3-({1-[4-(3-fluorophenyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}(1H-imidazol-2-ylmethyl)methylamine
4-chloro-2-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]phenol
1-[2-(2,3-dihydro-1H-isoindol-2-yl)-2-oxoethyl]-2-methyl-1,4-dihydroquinolin-4-one
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
N-(1-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}piperidin-4-yl)methanesulfonamide
4-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-1-(1H-1,2,3-triazole-5-carbonyl)piperidine
N,N-diethyl-1-[(1s,4s)-4-[3-(pyridin-3-yl)propanamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-[(1s,4s)-4-aminocyclohexyl]-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(1-{1-[(4-chloro-3-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
N-(2-methyl-1,3-benzothiazol-5-yl)morpholine-4-carboxamide
N-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}methanesulfonamide
N-benzyl-N-(cyclobutylmethyl)-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-(4-ethyl-1H-pyrazol-5-yl)-1-(2,4,5-trimethylbenzoyl)piperidine
1-[2-(1-methylpiperidin-2-yl)ethyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-{2-[4-(propan-2-yl)phenyl]pyrimidin-4-yl}pyrrolidin-3-ol