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(2R,3R,6R)-3-phenyl-5-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
6-(methoxymethyl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-4-amine
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]pyrazin-2-amine
4-(2-methoxyphenoxy)-1-(oxolan-3-ylmethyl)piperidine
(2S,4R)-4-amino-1-(2-butoxyacetyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-4-(1H-imidazol-1-yl)benzamide
1-[(3-chloro-4-fluorophenyl)methyl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
2-{1-methyl-4-[(2-methyl-1,3-oxazol-4-yl)methyl]-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl}acetic acid
5-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(ethyl)(oxolan-2-ylmethyl)amine
1-[(4-methoxyphenyl)methyl]-3-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-6-(morpholin-4-yl)pyrimidin-4-amine
4-[2-(4-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)ethyl]morpholine
2-cyclopentyl-N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)acetamide
(2R,6S)-4-{[1-butyl-2-(cyclohexanesulfonyl)-1H-imidazol-5-yl]methyl}-2,6-dimethylmorpholine
N-({5-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
4-(1-benzoxepine-4-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
4-{5-[(2E)-but-2-en-1-yl]-1,3,4-oxadiazole-2-carbonyl}-2-(4-fluorophenyl)morpholine
7-[4-(benzyloxy)butanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-(2-methylpropyl)-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}pyrrolidin-2-one
2-[ethyl(propan-2-yl)amino]-2-(2-methoxy-5-methylphenyl)acetic acid
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-3-(hydroxymethyl)piperidin-3-ol
[(3,4-dimethoxyphenyl)methyl](methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
2-(4-methoxypiperidin-1-yl)-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridine
1-({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)-4-(oxolane-2-carbonyl)piperazine
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
2-amino-8-hydroxy-4-(2-methyl-1H-imidazol-4-yl)-5H,6H-benzo[h]quinoline-3-carbonitrile
{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[2-(trifluoromethyl)phenyl]methyl}amine
7-(1-benzothiophen-3-yl)-4-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-indene-2-carboxamide
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-3-carboxamide
7-fluoro-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
N-(3-hydroxy-3-methylbutyl)-N,4-dimethyl-3-(2-oxoimidazolidin-1-yl)benzamide
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-(furan-2-yl)ethane-1,2-dione
7-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
2-(cyclopentylmethyl)-3-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-1-(2-methoxyethyl)-6-methyl-1,4-dihydropyridin-4-one
2-[4-(2-phenoxyethyl)piperazin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
4-(1-ethyl-1H-pyrazole-4-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-(phenoxymethyl)-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-1H-pyrazole-3-carboxamide
N-(1-carbamoylcyclopentyl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-N'-(4-fluorophenyl)ethanediamide
8-(1,3-benzoxazol-2-yl)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]-1,8-diazaspiro[4.5]decane
1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-4-(piperidin-1-yl)piperidine-4-carboxamide
7-(2-methoxyethyl)-2-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-(1-{1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxy-2-phenylacetamide
2-(2-chlorophenyl)-N-cyclobutyl-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-(1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperidine-4-carbonyl)morpholine
1-methoxy-8-(2,3,4,9-tetrahydro-1H-carbazole-1-carbonyl)-1,8-diazaspiro[4.5]decan-2-one
(3R,4R)-3-cyclobutyl-1-[(5-ethylpyridin-2-yl)methyl]-4-methylpyrrolidin-3-ol
2-{[(1-{[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine