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5-(3-chlorophenyl)-N-[2-(6-methylpyridin-2-yl)ethyl]-1,2,4-triazin-3-amine
7-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1-oxa-7-azaspiro[3.5]nonane
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
9-[(3-methylthiophen-2-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}acetamide
4-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
2-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-methyl-1H-1,2,3-benzotriazole-5-carboxamide
ethyl 1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-4-(2-phenylethyl)piperidine-4-carboxylate
4-chloro-N-[(3R,4S)-4-cyclopropyl-1-(3-methoxypropyl)pyrrolidin-3-yl]-1-ethyl-1H-pyrazole-5-carboxamide
1-{[(3S,4S)-1-[(4,5-dimethylfuran-2-yl)methyl]-3-hydroxypiperidin-4-yl]methyl}-3,3-diethylurea
5-{[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-amino-4-(3-methylthiophen-2-yl)-6-(trimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-(1,4-dithiepan-6-yl)-2-ethyl-2H-1,2,3,4-tetrazol-5-amine
N-[2-(methylsulfanyl)ethyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
2-benzyl-9-[(4-methoxypyridin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(pyrimidin-4-ylmethyl)amine
[(3R,4R)-4-(azepan-1-ylmethyl)-1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)pyrrolidin-3-yl]methanol
1-ethyl-3-[1-(2-hydroxyethyl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]-4,6-dimethyl-1,2-dihydropyridin-2-one
2-(4-chloro-2-methylphenoxy)-N-[(1s,4s)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexyl]propanamide
4-(azonan-1-ylmethyl)-N-(1,3,4-thiadiazol-2-yl)benzamide
2-[1-(2,3-dimethylquinoxalin-6-yl)-N-methylformamido]-2-(thiophen-2-yl)acetic acid
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
N-methyl-N-[(3-methylpyridin-2-yl)methyl]-1-[3-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
4-(3-hydroxy-3-methylbutyl)-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)benzamide
3-benzyl-6-(3-ethyl-1,2,4-oxadiazol-5-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)oxolane-3-carboxamide
ethyl[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl](oxan-4-ylmethyl)amine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,3-dimethyl-1H-pyrazole-4-carboxamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
4-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
6-chloro-N-(2-methoxyethyl)-1-methyl-N-(pyridin-3-ylmethyl)-1H-indole-2-carboxamide
3-methyl-N-[2-(6-oxo-3-phenyl-1,4,5,6-tetrahydropyridazin-1-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
(2S,4S)-4-amino-N,N-diethyl-1-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}pyrrolidine-2-carboxamide
2-(2-ethyl-1H-imidazol-1-yl)-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]ethan-1-one
ethyl({[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}){[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-[(1S,4S)-5-(2-methoxy-5-phenylphenyl)-6-oxo-2,5-diazabicyclo[2.2.1]heptan-2-yl]acetamide
7-fluoro-N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-2-methylquinoline-4-carboxamide
N-{[(2R)-1-ethylpyrrolidin-2-yl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
2-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-yl]-N-(3-fluorophenyl)-2-oxoacetamide
6-(2-chlorophenyl)-N-(2-hydroxyethyl)-N-methyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
(4aR,7aS)-1-propyl-4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
9-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-fluorophenyl)-N-(2-methoxyethyl)-2,2-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropane-1-carboxamide
4-(1,3-thiazol-2-ylmethyl)-3,4-dihydro-2H-1,4-benzothiazin-3-one
N-methyl-N-(quinolin-5-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-cyclopentyl-4-oxo-N-(2-phenylethyl)-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide