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2-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
2-(6-chloro-3-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline
(2S)-2-phenyl-2-({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethan-1-ol
2-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)-5,8-dimethylquinolin-4-ol
1-[(4aR,8aS)-6-[4-(trifluoromethyl)benzoyl]-decahydro-1,6-naphthyridin-1-yl]-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propan-1-one
7,7-dimethyl-2-[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
1-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1H-1,2,3-triazole
N-{4-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-oxobutyl}acetamide
1-[2-methoxy-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-3-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]urea
1-{2-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]phenyl}-3,5-dimethyl-1H-pyrazole
N-{3-[({1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}carbamoyl)amino]phenyl}acetamide
N-[(3-methylpyridin-4-yl)methyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-[1-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2,2-dimethylpropanamide
2-(dimethylamino)-N-(3-methoxypropyl)-4-methyl-N-[(4-methylphenyl)methyl]pyrimidine-5-carboxamide
1-methyl-2-{1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
N-[2-(dimethylamino)-2-(thiophen-2-yl)ethyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
N-(1,3-benzothiazol-2-ylmethyl)-4-[(2-methoxyethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-methyl-6-{1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-4-yl}pyrimidin-4-ol
2-(4-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)-1,3-benzoxazole
N-[3-(methylamino)propyl]-2-(4H-1,2,4-triazol-4-yl)benzamide
4-(piperidine-4-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(butylsulfanyl)-6-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyrimidin-4-amine
N-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-4-(pyrimidin-4-yl)piperidine-1-carboxamide
5-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-4-methyl-2-(pyridin-3-yl)pyrimidine
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-ethyl-N-[1-(4-methoxyphenyl)propan-2-yl]propanamide
2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidine
3-(3-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1H-pyrazol-3-yl}phenyl)-2,6-dimethylpyridine
1-[4-(hydroxymethyl)cyclohexanecarbonyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-[(1-cyclopentylpiperidin-3-yl)methyl]-2-methoxy-N-[2-(piperidin-1-yl)ethyl]acetamide
(3S,4R)-4-(hydroxymethyl)-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-3-ol
8-(1-ethyl-1H-pyrazole-5-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
6-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-4-amine
5-(1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
3-cyclohexyl-4-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1H-pyrazole
N-({6-[(3-fluorophenyl)methoxy]-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl}methyl)-2,2-dimethyloxan-4-amine
(3R,4S)-4-[methyl({[4-(methylsulfanyl)phenyl]methyl})amino]oxolan-3-ol
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
2-(4-fluoro-2-methoxyphenyl)-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetic acid
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-(4-methanesulfonylphenyl)ethan-1-one
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]benzamide
N-[4-({4-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)phenyl]acetamide
(4S)-3-[3-(2-methyl-1H-imidazol-1-yl)propyl]-4-phenyl-1,3-oxazolidin-2-one
(2R,3R)-3-{[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(quinolin-8-yl)pyridine-3-carbonitrile
N-(4-methylpentan-2-yl)-1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-amine
N-[2-(3,5-difluorophenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(adamantan-1-yl)-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methylacetamide
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-2-methylpropanamide
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(oxan-4-yl)ethyl]amine