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(3R,4S)-1-(1-methyl-1H-pyrazole-4-carbonyl)-4-propylpyrrolidin-3-amine
3-{2-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
methyl 4-({3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)benzoate
3-({1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]pyrrolidin-3-yl}methyl)benzoic acid
N-[(1R,3R)-3-aminocyclopentyl]-2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetamide
2-(2-{9-oxa-2-azaspiro[5.5]undecan-2-yl}-2-oxoethyl)-1,2-dihydroisoquinolin-1-one
2-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]pyrrolidin-2-yl}-1,3-thiazole
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl){pyrazolo[1,5-a]pyrimidin-3-ylmethyl}amine
2-[(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]-6-methylquinolin-4-ol
2-[(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)methyl]-4-methyl-1,2-dihydrophthalazin-1-one
3-(azepane-1-sulfonyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
2-fluoro-6-(4-phenyl-1H-imidazol-1-yl)benzamide
N4-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
3-({8-[2-(dimethylamino)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)benzonitrile
1'-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
N-[(3R,4S)-4-cyclopropyl-1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidin-3-yl]methanesulfonamide
N-[2-hydroxy-3-(4-methoxyphenoxy)propyl]-1,5-dimethyl-1H-indole-2-carboxamide
N-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-tert-butyl-1-methyl-1H-pyrazole-5-carboxamide
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3-(thiophene-2-carbonyl)piperidine
3-chloro-5-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
5-acetyl-2,4-dimethyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1H-pyrrole-3-carboxamide
(4aR,7aS)-1-(pyridin-4-ylmethyl)-4-(4,4,4-trifluorobutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]acetamide
N,2,3-trimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-indole-5-carboxamide
4-ethyl-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-1,2,3-thiadiazole-5-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)propanamide
4-(1-butyl-1H-imidazol-2-yl)-1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperidine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
1-(4-benzylpiperazin-1-yl)-3-[1-(thiophene-2-carbonyl)piperidin-3-yl]propan-1-one
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-[(2E)-3-phenylprop-2-en-1-yl]-4-[3-(1H-pyrazol-4-yl)benzoyl]piperazine
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}[1-(3-methylpyridin-2-yl)propan-2-yl]amine
4-(5-fluoropyrimidin-2-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-[4-(5-tert-butyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]quinazoline
3-ethyl-3-[(3S,4R)-4-hydroxyoxolan-3-yl]-1-(quinolin-8-yl)urea
2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-N-(oxan-2-ylmethyl)acetamide
N-methyl-5-{[methyl({5-methylpyrazolo[1,5-a]pyrimidin-7-yl})amino]methyl}pyrimidin-2-amine
2-(2-hydroxyethyl)-9-{[4-(1H-imidazol-1-yl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
2-(2-{[(1r,4r)-4-hydroxycyclohexyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
(2E)-3-(2-fluorophenyl)-1-{3-[5-phenyl-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}prop-2-en-1-one
6,8-dimethyl-2-({[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]amino}methyl)quinolin-4-ol
1-[(1,4-dimethyl-1H-pyrazol-5-yl)methyl]-4-(pyridin-3-ylmethyl)piperazine
4-({4-[4-(3-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)quinoline
2-{5-[1-(1H-imidazol-2-ylmethyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
(3S,4S)-4-cyclopropyl-1-[(4-methoxypiperidin-1-yl)sulfonyl]pyrrolidine-3-carboxylic acid
4-(3-methylphenoxy)-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidine
4-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
2-(2,3-dimethoxy-5-methylphenyl)-5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyridine