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4-methyl-2-[1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
methyl({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl})[1-(1,2-oxazol-3-yl)ethyl]amine
1-[(2R)-oxolane-2-carbonyl]-4-phenoxypiperidine-4-carboxylic acid
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]pyridine-3-carboxamide
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-methylpropanamide
1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
(2R,6S)-1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
3-[5-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]-1-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]urea
2-(5-tert-butyl-2H-1,2,3,4-tetrazol-2-yl)-N-{1-[(4-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}acetamide
N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}furan-3-carboxamide
2-(benzyloxy)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-{1-[4-(3-chlorophenyl)-5-({[3-(trifluoromethyl)phenyl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}furan-3-carboxamide
N-{2-[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperidin-3-yl]ethyl}acetamide
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluorobenzamide
1-(6-ethyl-2-methylpyrimidin-4-yl)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperidin-4-amine
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(2-methylpropyl)amine
2-(benzyloxy)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-benzyl-3-ethyl-1-(quinoline-8-carbonyl)-1,4-diazepan-5-one
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
N-{2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl}pyridin-3-amine
N-(1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-1-oxopropan-2-yl)-N-phenylmethanesulfonamide
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
6-[(3-chloro-4-hydroxyphenyl)methyl]-N-[2-(cyclohex-1-en-1-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-(furan-2-ylmethyl)piperidine
1-(dimethyl-1,3-thiazole-5-carbonyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
methyl({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})(1,3-thiazol-2-ylmethyl)amine
3-({[(2,4-dichloro-6-methylphenyl)methyl]amino}methyl)piperidin-3-ol
2-({[(3R,4R)-1-(1-benzothiophene-2-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-{4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-({[6-(4-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}(methyl)amino)-N-methylacetamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-ethyl-N-(oxolan-2-ylmethyl)-1,3-oxazole-4-carboxamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]ethan-1-one
{4-[(5-chloro-3-methoxy-2-propoxyphenyl)methyl]-1,4-oxazepan-6-yl}methanol
6-[2-(oxolan-3-yl)ethyl]-5,6-dihydro-1,6-naphthyridin-5-one
1-[2-(3-chlorophenyl)ethyl]-4-[(cyclopropylmethyl)amino]pyrrolidin-2-one
1-{2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}[1-(1H-indol-1-yl)propan-2-yl]amine
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
1,9-dimethyl-4-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
5-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-carbonyl)pyrazin-2-ol
3-methyl-N-[3-(5-methyl-4-{[2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamido]methyl}-1,3-oxazol-2-yl)phenyl]butanamide
1-{3-[3-(2-ethylphenoxy)azetidine-1-carbonyl]phenyl}-1H-pyrazole
5-methyl-1'-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(2-methylphenyl)-5-({3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)pyrimidine
N-[2-(cyclohexylsulfanyl)ethyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
N-cyclopropyl-1-(2-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
1-[4-(difluoromethoxy)-2-methylphenyl]-3-[3-(1H-1,2,3-triazol-1-yl)propyl]urea
5-{[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]methyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione