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6-(benzyloxy)-1-cyclohexyl-4-(pyridine-2-carbonyl)-1,4-diazepan-2-one
2-[1-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperidin-2-yl]acetic acid
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-[(1R,3R,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]propan-1-one
7-(cyclobutylmethyl)-2-(3-methylbut-2-enoyl)-2,7-diazaspiro[4.5]decan-6-one
7-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-(4-methylphenyl)-4-(2,3,6-trifluorobenzoyl)piperazin-2-one
8-{3-cyclopropyl-5-[(2S)-oxolan-2-yl]-1H-1,2,4-triazol-1-yl}quinoline
4-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}-1-oxaspiro[4.5]decan-2-one
4-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-6-methylpyrimidin-2-amine
(1R,4S)-2-[2-(3,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonyl]-2-azabicyclo[2.2.1]heptane
4-[4-(dimethylamino)phenyl]-3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
6-[(4aS,8aR)-1-(3-methoxypropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]pyrazine-2-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
1-(2-{1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]piperidin-4-yl}ethyl)pyrrolidin-2-one
N-[2-(2-fluorophenyl)ethyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
methyl 5-(3-oxo-3,4-dihydroquinoxaline-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-[(5-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]-3,3-dimethylurea
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(1-hydroxypropan-2-yl)acetamide
N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-(furan-2-yl)-4-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(1S,6R)-9-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
1-{6-[3-(1H-pyrazol-3-yl)phenyl]pyridin-2-yl}piperazine
5-chloro-6-oxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,6-dihydropyridine-3-carboxamide
4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]benzamide
3-(1,3-benzothiazol-2-yl)-N-[2-(N-methylmethanesulfonamido)ethyl]propanamide
3-(propan-2-yl)-N-{2-[(pyridin-2-ylmethyl)carbamoyl]phenyl}-1,2-oxazole-5-carboxamide
2-(4-chlorophenoxy)-1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
(1S,6R)-9-(4-cyclopentylpyrimidin-2-yl)-3-methyl-3,9-diazabicyclo[4.2.1]nonane
2-ethyl-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrimidine-5-carboxamide
1-{1'-[4-(ethylamino)pyrimidin-2-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-2-(dimethylamino)-2-(3-methylphenyl)acetamide
2-(3-methyl-1,2-oxazol-5-yl)-1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
(1R,2R,4R)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
N-[cyclopropyl(4-methoxyphenyl)methyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
6-methyl-2-{8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-3-carbonitrile
4-({[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)-2-methylbutan-2-ol
3,5,7-trimethyl-2-[3-(2-methylphenoxy)azetidine-1-carbonyl]-1H-indole
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
(3S,4R)-1-[3-(2-methoxyphenoxy)propyl]-4-methylpiperidine-3,4-diol
5-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-4-methyl-1,3-thiazole
3-{1-[2-methyl-2-(morpholin-4-yl)propanoyl]piperidin-3-yl}benzoic acid
N-{3-[4-(morpholin-4-ylmethyl)phenoxy]propyl}furan-2-carboxamide
3-{1-[2-(methylsulfanyl)phenyl]-N-(propan-2-yl)formamido}propanamide
N-methyl-2-({2-methylpyrido[2,3-d]pyrimidin-4-yl}amino)-2-phenylacetamide
9-(3-methoxy-2-methylbenzoyl)-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-(5-{[3-(4-fluoro-3-methylphenyl)-1-methyl-2-oxo-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-6-yl]methyl}thiophen-2-yl)acetamide
4-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
5-(2-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-oxoethyl)imidazolidine-2,4-dione
2-{[3-(aminomethyl)pyrrolidin-1-yl]methyl}-6,8-dimethylquinolin-4-ol