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N-[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]-2,6,8-trimethylquinoline-4-carboxamide
2,4-dimethoxy-5-[3-(1H-pyrazol-3-yl)phenyl]pyrimidine
(3R)-1-{3-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]benzenesulfonyl}pyrrolidin-3-ol
1-methyl-4-[3-(pyridin-3-yl)azetidine-1-carbonyl]-1,2-dihydroquinolin-2-one
[(4-fluorophenyl)[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl]dimethylamine
2-[(3,5-dichloropyridin-4-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-cyclobutyl-2-(1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-ethyl-8-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
ethyl 4-[(4-chlorophenyl)methyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-4-carboxylate
2-[2-(4-methyl-1,4-diazepan-1-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
4-[4-(3,4-difluorobenzoyl)piperidin-1-yl]-5-ethylpyrimidin-2-amine
2-(1H-1,3-benzodiazol-1-yl)-N-{2-[(4-methylphenyl)carbamoyl]ethyl}propanamide
3-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,5-dimethylphenyl)urea
2-[4-(2-ethylbutyl)piperazin-1-yl]pyridine-4-carbonitrile
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(dimethyl-1,2-oxazol-4-yl)acetamide
2-(6-methoxynaphthalen-2-yl)-4-(pyridin-4-yl)morpholine
5-(2H-1,3-benzodioxol-5-yl)-3-[3-(2-chlorophenyl)pyrrolidin-1-yl]-1,2,4-triazine
2-[4-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperazin-1-yl]pyrazine
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-methoxy-1-(pyridin-2-yl)ethyl]methylamine
4-[(2,4-diethoxy-3-methylphenyl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
1-(2-methylpropyl)-N-[2-(pyridin-3-yloxy)propyl]piperidin-4-amine
3-ethyl-1-methyl-N-(quinolin-5-yl)-1H-pyrazole-5-carboxamide
(2S)-2-amino-N-[3-(2,6-dimethylphenoxy)propyl]-3-methoxy-N-methylpropanamide
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
{5-[1-(2-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-1H-1,3-benzodiazol-2-yl}methanol
5-(2-propyl-1H-imidazol-1-yl)pyridin-3-amine
7,11-dimethyl-3-(5-propyl-1,3,4-oxadiazol-2-yl)-3,7,11-triazaspiro[5.6]dodecane
1-[3-(2-methoxypyridin-3-yl)-4-(morpholin-4-yl)phenyl]ethan-1-one
3-ethyl-8-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N,N-diethyl-1-{1-[(2-hydroxy-4-methoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
N-butyl-N-(furan-2-ylmethyl)-1-(pyrimidin-2-yl)piperidine-4-carboxamide
4-(2-phenylphenyl)-3-(pyridin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(1H-imidazol-4-yl)-1-{[3-(2-methoxyethoxy)phenyl]methyl}-4-phenyl-1H-imidazole
2-(4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
3-[4-(2-methoxybenzoyl)piperazine-1-carbonyl]-1,5,6-trimethyl-1,2-dihydropyridin-2-one
(2R,3R,6R)-3-(4-fluorophenyl)-5-(1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-[2-(2-fluorophenyl)ethyl]urea
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-2-ethylpyrimidine-5-carboxamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-3-(2-methoxyphenyl)-N-(oxolan-2-ylmethyl)propanamide
1-cycloheptyl-6-oxo-N-[2-(pyridin-4-yl)ethyl]piperidine-3-carboxamide
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
{1-[(5-cyclopropyl-4-phenyl-1H-imidazol-1-yl)methyl]cyclobutyl}methanol
1-[3,5-difluoro-4-(trifluoromethyl)phenyl]-3-(2,5-dihydroxy-2-methylpentyl)urea
9-(6-ethyl-2-methylpyrimidin-4-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methoxy-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyridine-3-carboxamide
1-(2-methylpropyl)-5-[(pyridin-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-(furan-2-ylmethyl)-3-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}urea
5-[4-(morpholin-4-yl)piperidine-1-carbonyl]-4-(trifluoromethyl)pyrimidin-2-amine
1-(oxolane-2-carbonyl)-N-(3-phenylprop-2-yn-1-yl)-N-propylpiperidine-4-carboxamide