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5-[(benzyloxy)methyl]-4-phenyl-1H-imidazole
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(2-phenylacetyl)pyrrolidin-3-yl]acetamide
3-phenyl-5-[1-(1H-pyrrol-1-yl)ethyl]-1H-1,2,4-triazole
(4aR,7aS)-1-benzyl-4-(2-hydroxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-{[2-(N-methylmethanesulfonamido)ethyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-4-phenylbutane-1,2-dione
4-[3-(3-chlorophenyl)pyrrolidine-1-carbonyl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-cyclobutylpiperidine
1'-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(oxolan-3-ylmethyl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
1-(2-methoxyethyl)-5-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]piperidin-2-one
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}cyclopropanesulfonamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
(2S,4R)-4-amino-N,N-diethyl-1-(9H-fluorene-9-carbonyl)pyrrolidine-2-carboxamide
(3aR,6aR)-2-(4-chloro-2-fluorobenzoyl)-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[1-(1-benzothiophen-2-ylmethyl)-4-hydroxypiperidin-4-yl]-N-(pyridin-2-ylmethyl)-1-benzofuran-2-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-3-(4-methylpiperazine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
N,N,2-trimethyl-3-[({3-[(5-methylpyridin-2-yl)amino]propyl}carbamoyl)amino]benzamide
(1-{1-[(1S,4S)-3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanol
2-(4-hydroxy-3-methoxyphenyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
8-[(dimethyl-1,3-thiazol-5-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[3-oxo-3-(pyrrolidin-1-yl)propyl]-1H-pyrazole-3-carboxamide
N-[1-(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-2-phenylethyl]-N-methylpyridine-2-carboxamide
4-{[2-(cyclopentyloxy)phenyl]methyl}-2-(pyridin-3-yl)morpholine
methyl 2-[1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octane-6-carbonyl]benzoate
4-(4-methanesulfonylphenyl)-2,6-dimethoxypyrimidine
3-(2-methoxyphenyl)-N-[(1-methylpiperidin-3-yl)methyl]benzamide
methyl 3-(3-methylthiophene-2-carbonyl)-9-[2-(morpholin-4-yl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-methyl-N-[1-(1-methyl-1H-imidazol-2-yl)butyl]-4-oxo-3,4-dihydrophthalazine-1-carboxamide
N-(isoquinolin-5-ylmethyl)-N-methyl-3-phenoxypropanamide
6-(2-methoxy-2-phenylacetyl)-1-[2-(piperidin-1-yl)ethyl]-3-(pyridin-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-[(3,5-difluorophenyl)methyl]-8-[1-(hydroxymethyl)cyclopropanecarbonyl]-2,8-diazaspiro[4.5]decan-3-one
N-cyclopentyl-N-[(5-methylthiophen-2-yl)methyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
4-{1-[3-(2-fluorophenoxy)azetidin-1-yl]-1-oxopropan-2-yl}-1,2-dihydrophthalazin-1-one
1-ethyl-2-({2-[(4-methoxyphenyl)methyl]morpholin-4-yl}methyl)-1H-1,3-benzodiazole
N-{[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
1-(propan-2-yl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidine-4-carboxamide
N-cyclopropyl-N'-(2-methylphenyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanediamide
5-methoxy-2-{[3-(4-phenylbenzoyl)piperidin-1-yl]methyl}-4H-pyran-4-one
N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-5,7-dimethyl-N-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-[(1-propyl-1H-imidazol-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
4-hydroxy-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
7-methyl-2-(1-methyl-1H-pyrazol-4-yl)-4-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}quinoline
(3S,9aR)-3-(cyclohexylmethyl)-8-(cyclopropylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-(4-{pyrazolo[1,5-a]pyrimidin-3-yl}phenyl)-1H-pyrazole
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-4-(1H-imidazol-1-yl)butan-1-one
3-[(oxan-4-ylmethyl)sulfamoyl]-N-(pyrrolidin-3-yl)benzamide
1-{1-[6-(2,6-dimethylphenyl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
8-(3-methoxypyrazin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one