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1-(cyclopent-1-ene-1-carbonyl)-3-[4-(naphthalen-1-yl)-1H-pyrazol-5-yl]piperidine
N-(1-propyl-1H-1,3-benzodiazol-5-yl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
N-(4-methoxy-2-methylphenyl)-3-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}propanamide
7-[(2-fluorophenyl)methyl]-2-(1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-{2-[1-(5-methoxypyrimidin-2-yl)piperidin-4-yl]ethyl}pyrrolidin-2-one
3-[(3,4-dimethoxypyridin-2-yl)methyl]-4,5-dimethyl-2,3-dihydro-1,3-oxazol-2-one
2-{3-[1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
N-(1H-imidazol-2-ylmethyl)-3-(3-methoxypiperidine-1-carbonyl)benzene-1-sulfonamide
9-[2-(ethanesulfonyl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1-methyl-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
1-[(4-chlorophenyl)methyl]-N-[3-(3-hydroxypiperidin-1-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
3-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-(2,3-dihydro-1H-inden-5-yl)urea
2-[3-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)propyl]-5-(4-fluorophenyl)-2H-1,2,3,4-tetrazole
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1,5-dimethyl-1H-indazole-3-carboxamide
1-methyl-N-[3-(pyridin-2-yl)propyl]-1H-1,2,3-benzotriazole-5-carboxamide
1-[3-(3-chlorophenyl)phenyl]-3-{[4-(dimethylamino)oxan-4-yl]methyl}urea
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-2-methyl-5-(2-methyl-1,3-oxazol-5-yl)benzene-1-sulfonamide
5-({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}(methyl)carbamoyl)thiophene-2-carboxylic acid
(4aR,7aS)-1-acetyl-4-{2-[(2-methylphenyl)sulfanyl]acetyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4S)-4-amino-1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-N-ethylpyrrolidine-2-carboxamide
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
5-(2-fluoro-4-methoxyphenyl)-4-phenyl-1-[2-(propan-2-yloxy)ethyl]-1H-imidazole
{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
N-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)-N-methylmethanesulfonamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)pyrrolidin-3-yl]methanol
(3S,4S)-1-[4-(aminomethyl)benzoyl]-4-(naphthalen-2-yl)piperidin-3-ol
8-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
6-methyl-4-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]quinoline
4-(1-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-1H-imidazol-2-yl)-N,N-dimethylaniline
5-{[4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}quinoxaline
4-ethyl-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-methyl-1,3-thiazole-5-carboxamide
3-{[1-(1-methoxypropan-2-yl)piperidin-4-yl]oxy}-N-(pyridin-3-ylmethyl)benzamide
N2-benzyl-N2,7,7-trimethyl-N5-[(1-methyl-1H-pyrazol-4-yl)methyl]-5,6,7,8-tetrahydroquinazoline-2,5-diamine
({5-[(4-chlorophenyl)sulfanyl]furan-2-yl}methyl)(2-methanesulfonylethyl)amine
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[(2-ethoxypyridin-3-yl)methyl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
2-[3-({[2-(1H-imidazol-1-yl)ethyl](methyl)amino}methyl)phenyl]-6-(oxan-4-yl)-3,4-dihydropyrimidin-4-one
N-(2-methoxyethyl)-1-[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
2-{[(2S)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]methyl}-1H-1,3-benzodiazole
4-[(4-chloro-3-fluorophenyl)methyl]-3-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-2-one
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)acetamide
N-(2-methoxyphenyl)-1-{2-[2-(trifluoromethyl)benzenesulfonamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
1-[(4-methoxyphenyl)methyl]-4-[2-(thiophen-3-yl)acetyl]piperazin-2-one
6,7-dimethoxy-2-(2-methylquinolin-5-yl)quinazolin-4-amine
(4aR,7aS)-1-cyclobutanecarbonyl-4-(3-hydroxypyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(propylsulfanyl)ethyl]piperidin-4-amine
2-tert-butyl-N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-4-hydroxypyrimidine-5-carboxamide