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2,3-dimethyl-6-[3-(pyridin-3-yl)propanoyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-(2-acetamidophenyl)-2-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]acetamide
1-[1-(3-hydroxypropyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-ethyl-3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
4-methyl-2-(propan-2-yl)-5-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]-1,3-thiazole
[2-({4-[1-(prop-2-en-1-yl)pyrrolidine-2-carbonyl]piperazin-1-yl}methyl)phenyl]methanol
4-(1-benzyl-1H-imidazol-2-yl)-1-(2-fluorobenzoyl)piperidine
4-[(4-chlorophenyl)methyl]-1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]piperidine-4-carboxylic acid
N-[(3S,4R)-1-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
N-cyclopropyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-2-(trifluoromethyl)benzamide
3-butyl-4-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-1-methylpiperazin-2-one
1-cyclopentyl-4-(2-ethylpyrimidine-5-carbonyl)-1,4-diazepane
2-[2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-5,6-dimethylpyridine-3-carbonitrile
2-{[(3aS,6aS)-5-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-octahydropyrrolo[3,4-b]pyrrol-1-yl]methyl}-1-methyl-1H-imidazole
N-[2-(pyridin-3-yl)phenyl]cyclopropanecarboxamide
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-4-(trifluoromethyl)pyrimidin-2-amine
3-ethoxy-2-hydroxy-S-[3-(piperazine-1-carbonyl)phenyl]propane-1-sulfonamido
3-{[4-(4-acetylphenyl)piperazin-1-yl]methyl}-N-butyl-N-methylimidazo[1,2-a]pyridine-2-carboxamide
5-methyl-N,N-bis(prop-2-en-1-yl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-[3-(pyridin-4-yl)-5-[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-1,2,4-triazol-1-yl]butan-2-ol
5-[4-hydroxy-1-(3-methylbut-2-en-1-yl)piperidin-4-yl]-N-methyl-N-(quinolin-6-ylmethyl)-1-benzofuran-2-carboxamide
4-methyl-5-{3-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-phenoxypropanamide
2-(2-{[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]methyl}-1H-pyrrol-1-yl)pyrimidine
5-(butan-2-yl)-1-(2-methylpropyl)-1H,4H-pyrazolo[3,4-d]imidazole
7-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-oxa-7-azaspiro[4.5]decane
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}piperidin-2-one
N-[2-(3-methoxyphenyl)ethyl]-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-({1-[6-(1,4-oxazepan-4-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-N-(propan-2-yl)-4-(1H-pyrazol-3-yl)benzamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-(propan-2-yl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl][(2,2-dimethyloxan-4-yl)methyl]methylamine
3-(1-ethyl-1H-imidazol-2-yl)-1-(4-fluorobenzenesulfonyl)piperidine
2-methyl-4-{[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-imidazole
{[(3S,4R)-1-(1,3-benzothiazol-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
ethyl(methyl)[(5-{3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]amine
2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-4-(1H-1,2,3,4-tetrazol-1-yl)phenol
N-[2-(dimethylamino)ethyl]-5-(3,3-dimethylbutanoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-({[(2-methoxyphenyl)methyl](prop-2-en-1-yl)amino}methyl)benzonitrile
5-[4-(adamantan-2-yl)piperazin-1-yl]-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
(3S,4S)-1-[2-(6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-[4-(5-tert-butyl-1H-pyrazol-3-yl)-7-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl]propanamide
5-(4-methoxyphenyl)-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
8-(3-carboxy-5-methoxybenzoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-{[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
4-methylphenyl (7S,9aR)-7-[(4-methoxyphenyl)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
7-(3-chlorophenyl)-4-[2-(5-methyl-1H-pyrazol-1-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
9-(cyclopropylmethyl)-1-methyl-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
4-phenyl-N-{1-[1-(thiophene-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
1-ethyl-N-[(4-fluorophenyl)methyl]-3,5-dimethyl-N-(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide